SCHEMBL7094941

SCHEMBL7094941

c1cc2c(cc1OC[C@@H]1CO1)OCO2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
TP53 P04637 4/20 0.59
TSHR P16473 3/20 0.59
CYP3A4 P08684 3/20 0.59
HIF1A Q16665 2/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
MAOB P27338 8/20 0.55
TDP1 Q9NUW8 2/20 0.51
MAOA P21397 4/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
MAPT P10636 2/20 0.49
HPGD P15428 2/20 0.49
CYP1A2 P05177 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
PPARG P37231 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
PKM P14618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7979964 1.00 ALDH1A1 (0.59) ALDH1A1TP53TSHRCYP3A4HIF1A
SCHEMBL5515785 1.00 ALDH1A1 (0.59) ALDH1A1TP53TSHRCYP3A4HIF1A
SCHEMBL8151638 0.83 ALDH1A1 (0.62) ALDH1A1TP53TSHRCYP3A4HIF1A
SCHEMBL983383 0.81 MAOB (0.57) ALDH1A1TP53CYP3A4SMN1; SMN2MAOB
SCHEMBL6782574 0.79 MAOB (0.65) ALDH1A1SMN1; SMN2MAOBMAOANPC1
SCHEMBL985688 0.79 MAOB (0.54) ALDH1A1TP53CYP3A4MAOBTDP1
SCHEMBL107322 0.78 MAOB (0.83) ALDH1A1TSHRCYP3A4MAOBTDP1
SCHEMBL1715242 0.78 ALDH1A1 (0.71) ALDH1A1TP53TSHRCYP3A4HIF1A
SCHEMBL21094081 0.78 TDP1 (0.79) ALDH1A1TP53TSHRCYP3A4HIF1A
SCHEMBL20677146 0.78 TDP1 (0.79) ALDH1A1TP53TSHRCYP3A4HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11773086-B2 Fungal modulators TRUSTEES OF BOSTON UNIVERSITY (US) 2023-10-03 US disclosed
US-11773086-B2 Fungal modulators TRUSTEES OF BOSTON UNIVERSITY (US) 2023-10-03 US disclosed
US-20220064152-A1 NOVEL FUNGAL MODULATORS TRUSTEES OF BOSTON UNIVERSITY (US) 2022-03-03 US disclosed
US-6605618-B2 Antidiabetic agents; hypoglycemic agents; anticholesterol agents; side effect reduction WYETH 2003-08-12 US disclosed
US-20030018045-A1 Heterocyclic beta-3 adrenergic receptor agonists WYETH (US) 2003-01-23 US disclosed
US-6458817-B1 AROMATIC SUBSTITUTED SUFURE OR SULFOXIDE OR SULFONE DERIVATIVES CONTAINING SECONDAY AMINE AND HYDROXY GROUPS ARE USEFUL IN TREATNG METABOLIC DISORDERS MEDIATED BY INSULIN RESISTANCE OR HYPERGLYCEMIA IN MAMMALS WYETH 2002-10-01 US disclosed
US-6451814-B1 SUBSTITUTED 4-((4-AMINO-5-HYDROXYPHENYL)-OXY-)PIPERIDINE ANALOGS; METABOLIC DISORDERS; ANTIDIABETIC AGENTS; ATHERO-SCLEROSIS, GASTROINTESTINAL DISORDERS, GLAUCOMA, NEUROGENETIC INFLAMMATION, OCULAR HYPERTENSION AND FREQUENT URINATION WYETH 2002-09-17 US disclosed
US-20020040023-A1 Substituted arylsulfides, arylsulfoxides and arylsulfones as beta-3 adrenergic receptor agonists AMERICAN HOME PRODUCTS CORPORATION (US) 2002-04-04 US disclosed
US-20020028832-A1 Heterocyclic beta-3 adrenergic receptor agonists AMERICAN HOME PRODUCTS CORPORATION (US) 2002-03-07 US disclosed
WO-2001017993-A1 ALKYLPIPERIDI NYLBENZO [D] ISOXAZOLE DERIVATIVES HAVING PSYCHOTROPIC ACTIVITY, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND A PROCESS FOR THE PREPARATION OF THE ACTIVE INGREDIENT EGIS Gyógyszergyár Rt. (HU) 2001-03-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030018045-A1 Heterocyclic beta-3 adrenergic receptor agonists ADRB2, ADRB1, ADRB3 ALDH1A1 725/4885TP53 4790/4885TSHR 603/4885
US-11773086-B2 Fungal modulators ABCB11, ABCB1, ABCC1 ALDH1A1 3436/4885TP53 1316/4885TSHR 4863/4885
US-20020040023-A1 Substituted arylsulfides, arylsulfoxides and arylsulfones as beta-3 adrenergic receptor agonists ADRB1, ADRB3, GPR119 ALDH1A1 602/4885TP53 4670/4885TSHR 296/4885
US-20020028832-A1 Heterocyclic beta-3 adrenergic receptor agonists ADRB1, ADRB3, ADRB2 ALDH1A1 524/4885TP53 4644/4885TSHR 552/4885
US-20220064152-A1 NOVEL FUNGAL MODULATORS ABCB11, ABCB1, ABCC1 ALDH1A1 3676/4885TP53 1931/4885TSHR 4863/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.