SCHEMBL7095121

SCHEMBL7095121

COc1cc2c(cc1OCCN1CCN(C(=O)OC(C)(C)C)CC1)NCC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP2C19 P33261 1/20 0.42
EHMT2 Q96KQ7 2/20 0.42
NSD2 O96028 1/20 0.42
TLR9 Q9NR96 2/20 0.41
TLR7 Q9NYK1 2/20 0.41
CFTR P13569 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
DRD3 P35462 2/20 0.40
KMT5A Q9NQR1 1/20 0.40
MAPK1 P28482 1/20 0.40
EPHX2 P34913 2/20 0.39
DRD2 P14416 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
GPR4 P46093 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7092953 0.81 EHMT2 (0.56) EHMT2
SCHEMBL8306947 0.80 MAPK1 (0.45) ALDH1A1CYP2C9ALOX15CYP2C19TLR9
SCHEMBL7097649 0.80 EHMT2 (0.55) EHMT2
SCHEMBL7094017 0.78 SYK (0.52) ALDH1A1EHMT2GAATSHRMAPK1
SCHEMBL7005111 0.76 DRD3 (0.48) RXFP1ALDH1A1EHMT2NSD2CFTR
SCHEMBL7011905 0.73 ALDH1A1 (0.53) RXFP1ALDH1A1MAPTDRD3DRD2
SCHEMBL19479118 0.72 DRD3 (0.70) ALDH1A1DRD3DRD2
SCHEMBL1667304 0.71 NSD2 (0.49) ALDH1A1EHMT2NSD2TLR9TLR7
SCHEMBL3196231 0.71 DRD3 (0.50) RXFP1ALDH1A1TLR9TLR7DRD3
SCHEMBL25221277 0.71 ALDH1A1 (0.52) ALDH1A1CYP2C9ALOX15CYP2C19GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309551-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2003-05-14 EP disclosed
WO-2002014273-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-02-21 WO disclosed