SCHEMBL7095589

SCHEMBL7095589

CC(=O)Oc1c(C)cc(OCCN2CCNCC2)c(C)c1C

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
KDM4E B2RXH2 6/20 0.47
ALDH1A1 P00352 4/20 0.47
GAA P10253 1/20 0.47
TP53 P04637 1/20 0.47
POLB P06746 1/20 0.41
ALOX5 P09917 1/20 0.41
P2RY12 Q9H244 1/20 0.41
TDP1 Q9NUW8 3/20 0.40
CREBBP Q92793 1/20 0.40
MAPT P10636 1/20 0.40
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7094471 0.80 ALOX5 (0.39) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL7096822 0.74 HTT (0.45) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL9015990 0.73 HTT (0.44) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL9053303 0.73 HTT (0.44) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL8005768 0.73 MEN1 (0.52) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL688109 0.72 THRA (0.46) MEN1KMT2AALDH1A1POLBALOX5
SCHEMBL9015951 0.71 MEN1 (0.55) MEN1KMT2AKDM4EALDH1A1
SCHEMBL2910532 0.70 POLB (0.62) KMT2AKDM4EALDH1A1GAATP53
SCHEMBL1495906 0.70 CREBBP (0.55) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL8669046 0.70 HTR1A (0.64) MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1361875-A2 NOVEL HETEROCYCLIC AMIDE DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS Aventis Pharmaceuticals Inc. (US) 2003-11-19 EP claimed
WO-2002066469-A2 NOVEL HETEROCYCLIC AMIDE DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS AVENTIS PHARMACEUTICALS INC. (US) 2002-08-29 WO claimed
EP-0901469-B1 ARYLALKYLPIPERAZINE COMPOUNDS AS ANTIOXIDANTS UNIV MONASH (AU) 2003-08-27 EP disclosed
US-6232314-B1 SUCH AS 1-(2-(4-CHLOROPHENYL)-2-HYDROXY)ETHYL-4-(3,5-BIS(1,1-DIMETHYLETHYL)-4 -HYDROXYPHENYL)METHYLPIPERAZINE; USED TO TREAT STROKE, CARDIAC ARREST, ISCHAEMIA, HYPOXIA, HYPOGLYCAEMIA, EPILEPSY, AND AMYOTROPHIC LATERAL SCLEROSIS MONASH UNIVERSITY (AU) 2001-05-15 US disclosed