SCHEMBL7097138

SCHEMBL7097138

CS(=O)(=O)c1c(=O)n(Cc2ccccc2)c(=O)n2cc(C(=O)O)sc12

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 15/20 0.55
MMP13 P45452 1/20 0.42
ALDH1A1 P00352 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7103846 0.90 TRPA1 (0.45) TRPA1
SCHEMBL7099747 0.89 TRPA1 (0.45) TRPA1MMP13ALDH1A1
SCHEMBL7167986 0.87 TRPA1 (0.43) TRPA1
SCHEMBL7097571 0.85 TRPA1 (0.60) TRPA1MMP13ALDH1A1
SCHEMBL5957285 0.83 TRPA1 (0.76) TRPA1MMP13
SCHEMBL7152830 0.81 TRPA1 (0.65) TRPA1ALDH1A1
SCHEMBL6514529 0.80 TRPA1 (0.59) TRPA1
SCHEMBL5957429 0.75 TRPA1 (0.73) TRPA1MMP13ALDH1A1
SCHEMBL6236419 0.75 TRPA1 (0.63) TRPA1
SCHEMBL6233188 0.75 TRPA1 (0.58) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362054-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP disclosed
WO-2002064599-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed