SCHEMBL7103846

SCHEMBL7103846

CS(=O)(=O)c1c(=O)n(Cc2ccc(Br)cc2)c(=O)n2cc(C(=O)O)sc12

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 13/20 0.45
POLB P06746 1/20 0.39
ERCC5 P28715 2/20 0.38
FEN1 P39748 2/20 0.38
PTGS2 P35354 1/20 0.37
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7097138 0.90 TRPA1 (0.55) TRPA1
SCHEMBL7099747 0.88 TRPA1 (0.45) TRPA1ERCC5FEN1
SCHEMBL7167986 0.87 TRPA1 (0.43) TRPA1ERCC5FEN1PTGDR2
SCHEMBL6239555 0.84 TRPA1 (0.62) TRPA1POLBERCC5FEN1
SCHEMBL6514529 0.80 TRPA1 (0.59) TRPA1ERCC5FEN1MAPK8PTGDR2
SCHEMBL7097571 0.76 TRPA1 (0.60) TRPA1
SCHEMBL7152830 0.75 TRPA1 (0.65) TRPA1
SCHEMBL6233188 0.74 TRPA1 (0.58) TRPA1
SCHEMBL6235332 0.74 TRPA1 (0.72) TRPA1POLB
SCHEMBL5957285 0.74 TRPA1 (0.76) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362054-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP disclosed
WO-2002064599-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed