SCHEMBL7099747

SCHEMBL7099747

CS(=O)(=O)c1c(=O)n(Cc2cccc(Br)c2)c(=O)n2cc(C(=O)O)sc12

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 13/20 0.45
ERCC5 P28715 2/20 0.41
FEN1 P39748 2/20 0.41
MAPK1 P28482 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HIF1A Q16665 1/20 0.38
LMNA P02545 1/20 0.36
PRNP P04156 1/20 0.36
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7097138 0.89 TRPA1 (0.55) TRPA1ALDH1A1MMP13
SCHEMBL7103846 0.88 TRPA1 (0.45) TRPA1ERCC5FEN1
SCHEMBL6237698 0.86 TRPA1 (0.60) TRPA1ERCC5FEN1MAPK1MEN1
SCHEMBL7167986 0.79 TRPA1 (0.43) TRPA1ERCC5FEN1
SCHEMBL7097571 0.75 TRPA1 (0.60) TRPA1ALDH1A1MMP13
SCHEMBL6238345 0.73 TRPA1 (0.62) TRPA1FEN1LMNA
SCHEMBL6236419 0.73 TRPA1 (0.63) TRPA1
SCHEMBL5957285 0.73 TRPA1 (0.76) TRPA1MMP13
SCHEMBL6239555 0.73 TRPA1 (0.62) TRPA1ERCC5FEN1
SCHEMBL6514529 0.72 TRPA1 (0.59) TRPA1ERCC5FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362054-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP disclosed
WO-2002064599-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed