SCHEMBL7167986

SCHEMBL7167986

CS(=O)(=O)c1c(=O)n(Cc2ccc(C#N)cc2)c(=O)n2cc(C(=O)O)sc12

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 13/20 0.43
FEN1 P39748 1/20 0.40
AR P10275 1/20 0.38
ERCC5 P28715 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
GAA P10253 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7097138 0.87 TRPA1 (0.55) TRPA1
SCHEMBL7103846 0.87 TRPA1 (0.45) TRPA1FEN1ERCC5PTGDR2
SCHEMBL5957391 0.85 TRPA1 (0.59) TRPA1FEN1ARERCC5
SCHEMBL7150079 0.84 TRPA1 (0.62) TRPA1
SCHEMBL7099747 0.79 TRPA1 (0.45) TRPA1FEN1ERCC5
SCHEMBL6514529 0.77 TRPA1 (0.59) TRPA1FEN1ERCC5PTGDR2
SCHEMBL7097571 0.76 TRPA1 (0.60) TRPA1
SCHEMBL6236549 0.74 TRPA1 (0.57) TRPA1FEN1ERCC5
SCHEMBL7038890 0.73 MMP13 (0.46) TRPA1FEN1ARPTGDR2GAA
SCHEMBL7152830 0.72 TRPA1 (0.65) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362054-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP disclosed
WO-2002064599-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed