SCHEMBL7097571

SCHEMBL7097571

C#CCNC(=O)c1cn2c(=O)n(Cc3ccccc3)c(=O)c(S(C)(=O)=O)c2s1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 15/20 0.60
MMP13 P45452 1/20 0.37
ALOX15 P16050 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KDM5B Q9UGL1 1/20 0.35
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5957424 0.86 TRPA1 (0.79) TRPA1MMP13TP53
SCHEMBL7097138 0.85 TRPA1 (0.55) TRPA1MMP13ALDH1A1
SCHEMBL7152830 0.83 TRPA1 (0.65) TRPA1ALDH1A1TP53
SCHEMBL7150079 0.76 TRPA1 (0.62) TRPA1ALDH1A1
SCHEMBL7103846 0.76 TRPA1 (0.45) TRPA1
SCHEMBL7167986 0.76 TRPA1 (0.43) TRPA1
SCHEMBL7099747 0.75 TRPA1 (0.45) TRPA1MMP13ALDH1A1
SCHEMBL5957632 0.75 TRPA1 (1.00) TRPA1TP53
SCHEMBL5957359 0.72 TRPA1 (1.00) TRPA1TP53
SCHEMBL5957636 0.71 TRPA1 (1.00) TRPA1ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362054-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP disclosed
WO-2002064599-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed