SCHEMBL7097152

SCHEMBL7097152

COc1cccc(OC)c1C=CC(=O)c1ccccc1N

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 5/20 0.63
ABCB1 P08183 1/20 0.57
MAPT P10636 3/20 0.56
CYP1A1 P04798 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
MAOB P27338 3/20 0.52
AR P10275 2/20 0.52
NR1H4 Q96RI1 1/20 0.52
AURKA O14965 1/20 0.48
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 2/20 0.47
HPGD P15428 2/20 0.47
RCE1 Q9Y256 1/20 0.47
CFTR P13569 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
HTT P42858 1/20 0.46
RECQL P46063 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7102181 0.87 ABCG2 (0.63) ABCG2ABCB1MAPTAURKAMEN1
SCHEMBL7100046 0.85 AR (0.72) ABCG2MAPTCYP1A1CYP1A2CYP2D6
SCHEMBL8102696 0.84 MAOB (0.74) ABCG2ABCB1MAPTCYP2D6MAOB
SCHEMBL8102695 0.84 MAOB (0.74) ABCG2ABCB1MAPTCYP2D6MAOB
SCHEMBL7096835 0.83 NFE2L2 (0.63) MAPTCYP1A1CYP1A2CYP2D6MAOB
SCHEMBL7099965 0.80 KDM4E (0.63) ABCG2ABCB1MAPTCYP1A1CYP1A2
SCHEMBL7098150 0.80 ABCG2 (0.62) ABCG2MAPTMAOBARNR1H4
SCHEMBL29211623 0.79 ABCG2 (0.66) ABCG2ABCB1MAPTCYP2D6MAOB
SCHEMBL27907245 0.79 ABCG2 (0.74) ABCG2ABCB1MAPTCYP1A2MAOB
SCHEMBL27907246 0.79 ABCG2 (0.74) ABCG2ABCB1MAPTCYP1A2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003097577-A1 CHEMICAL COMPOUND CONSISTING OF A NITROGENOUS CHALCONE DERIVATIVE, METHOD OF PRODUCING ONE SUCH CHEMICAL COMPOUND AND FILTERING AND/OR COSMETIC COMPOSITION CONTAINING SAME SYNTH'E163 (SOCIETE ANONYME) (FR) 2003-11-27 WO claimed
WO-2003097577-A1 CHEMICAL COMPOUND CONSISTING OF A NITROGENOUS CHALCONE DERIVATIVE, METHOD OF PRODUCING ONE SUCH CHEMICAL COMPOUND AND FILTERING AND/OR COSMETIC COMPOSITION CONTAINING SAME SYNTH'E163 (SOCIETE ANONYME) (FR) 2003-11-27 WO disclosed