SCHEMBL7097969

SCHEMBL7097969

O=C(NCCCCCCNC(=S)Nc1ccncc1)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.64
JAK2 O60674 1/20 0.57
TYK2 P29597 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
ALDH1A1 P00352 3/20 0.56
CA9 Q16790 2/20 0.56
CA1 P00915 1/20 0.56
GAA P10253 1/20 0.56
LMNA P02545 1/20 0.55
HPGD P15428 1/20 0.55
MAPK1 P28482 1/20 0.55
NAAA Q02083 2/20 0.55
HDAC3 O15379 2/20 0.54
HDAC1 Q13547 2/20 0.54
HDAC4 P56524 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC10 Q969S8 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7966915 0.84 CA9 (0.54) EPHX1ALDH1A1CA9LMNAHTT
SCHEMBL7104425 0.83 HDAC4 (0.63) ALDH1A1MAPK1HDAC3HDAC1HDAC4
SCHEMBL8915063 0.82 CA9 (0.58) ALDH1A1CA9GAALMNARAB9A
SCHEMBL7904143 0.81 KMT2A (0.71) ALDH1A1CA9GAALMNAMAPK1
SCHEMBL7901763 0.81 KMT2A (0.71) ALDH1A1CA9GAALMNAMAPK1
SCHEMBL8915308 0.81 CA9 (0.60) ALDH1A1CA9GAALMNARAB9A
SCHEMBL8916068 0.79 L3MBTL1 (0.56) ALDH1A1CA9GAALMNAHPGD
SCHEMBL8917236 0.79 L3MBTL1 (0.56) ALDH1A1CA9GAALMNAHPGD
SCHEMBL8916892 0.79 L3MBTL1 (0.56) ALDH1A1CA9GAALMNAHPGD
SCHEMBL8916496 0.79 L3MBTL1 (0.56) ALDH1A1CA9GAALMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984938-B1 CYANOGUANIDINES AS CELL PROLIFERATION INHIBITORS LEO PHARMA AS WITH SECONDARY N (DK) 2003-09-10 EP disclosed
US-6346541-B1 ANTITUMOR AND ANTICARCINOGENIC AGENTS FOR BREAST, LUNG, AND SKIN CANCER LEO PHARMACEUTICAL PRODUCTS LTD. A/S (DK) 2002-02-12 US disclosed