SCHEMBL7100301

SCHEMBL7100301

C=C1C[C@H](O)[C@@]2(C)CCC3c4ccc(N(C)S(=O)(=O)O)cc4CCC3[C@H]12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.47
ABCC4 O15439 1/20 0.47
STS P08842 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ESR1 P03372 5/20 0.44
HSD17B10 Q99714 4/20 0.44
LMNA P02545 4/20 0.44
ESR2 Q92731 3/20 0.44
TSHR P16473 2/20 0.44
PGR P06401 2/20 0.44
AR P10275 2/20 0.44
SLC6A3 Q01959 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HIF1A Q16665 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SLC22A1 O15245 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5266573 0.84 LMNA (0.44) ABCC1ABCC4STSKDM4EESR1
SCHEMBL5266242 0.84 LMNA (0.44) ABCC1ABCC4STSKDM4EESR1
SCHEMBL5266311 0.83 ABCC4 (0.43) ABCC1ABCC4STSKDM4EESR1
SCHEMBL5267416 0.83 ABCC4 (0.43) ABCC1ABCC4STSKDM4EESR1
SCHEMBL7098854 0.82 ABCC4 (0.55) ABCC1ABCC4STSKDM4EESR1
SCHEMBL7097126 0.82 ABCC1 (0.48) ABCC1ABCC4STSKDM4EESR1
SCHEMBL6636478 0.82 ABCC1 (0.48) ABCC1ABCC4STSKDM4EESR1
SCHEMBL5675177 0.82 ESR1 (0.64) STSESR1HSD17B10LMNAESR2
SCHEMBL7147482 0.82 ESR1 (0.64) STSESR1HSD17B10LMNAESR2
SCHEMBL8623796 0.80 LMNA (0.67) ABCC1ABCC4STSKDM4EESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775156-B1 PHARMACEUTICAL COMPOSITIONS CONTAINING ESTRA-1,3,5(10)-TRIENE DERIVATIVES JENAPHARM GMBH (DE) 2003-09-03 EP claimed