SCHEMBL7100441

SCHEMBL7100441

COc1ccc2ncc(CO)c(CC[CH]F)c2c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 9/20 0.40
MTNR1A P48039 8/20 0.40
KDM4E B2RXH2 3/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ROCK2 O75116 1/20 0.38
ALDH1A1 P00352 2/20 0.38
F2 P00734 1/20 0.38
GLA P06280 1/20 0.38
HPGD P15428 1/20 0.38
LMNA P02545 1/20 0.38
CYP19A1 P11511 1/20 0.38
HTR1A P08908 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
CYP1A2 P05177 1/20 0.36
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27580125 0.84 MTNR1B (0.42) MTNR1BMTNR1AKDM4EMAPK1NPSR1
SCHEMBL2010360 0.76 LMNA (0.44) MTNR1BMTNR1AKDM4EMAPK1NPSR1
SCHEMBL11070962 0.76 KDM4E (0.44) MTNR1BMTNR1AKDM4EMAPK1NPSR1
SCHEMBL2533923 0.75 KCNH2 (0.46) KDM4EMAPK1NPSR1ROCK2LMNA
SCHEMBL6267955 0.73 KCNH2 (0.48) LMNAKCNH2
SCHEMBL2011583 0.72 LMNA (0.43) MTNR1BMTNR1AKDM4EMAPK1NPSR1
SCHEMBL7100445 0.72 ROCK2 (0.41) MTNR1BMTNR1AKDM4EMAPK1NPSR1
SCHEMBL7065988 0.71 PLA2G2A (0.43) MTNR1BMTNR1AKDM4EMAPK1NPSR1
SCHEMBL7066589 0.71 ICAM1 (0.41) MTNR1BMTNR1AKDM4EMAPK1NPSR1
SCHEMBL14250570 0.70 PTGS1 (0.42) MTNR1BMTNR1AKDM4EMAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337529-A2 HETEROCYCLYLALKYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND COMPOSITIONS CONTAINING SAME Aventis Pharma S.A. (FR) 2003-08-27 EP disclosed
WO-2002040474-A2 HETEROCYCLYLALKYL PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIMICROBIAL AGENTS AVENTIS PHARMA S.A. (FR) 2002-05-23 WO disclosed