SCHEMBL7100445

SCHEMBL7100445

[CH2]CC(F)c1c(CO)cnc2ccc(OC)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.41
MTNR1A P48039 6/20 0.39
MTNR1B P49286 6/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
F2 P00734 1/20 0.39
GLA P06280 1/20 0.39
HPGD P15428 1/20 0.39
LMNA P02545 1/20 0.39
CYP19A1 P11511 1/20 0.38
HTR1A P08908 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
GABRA1 P14867 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11070962 0.77 KDM4E (0.44) ROCK2MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL27580125 0.77 MTNR1B (0.42) ROCK2MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL7066589 0.74 ICAM1 (0.41) ROCK2MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL28160791 0.73 ALDH1A1 (0.43) ROCK2MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL7461216 0.72 ADRA1A (0.50) ROCK2MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL7065988 0.72 PLA2G2A (0.43) ROCK2MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL7100441 0.72 MTNR1B (0.40) ROCK2MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL2544860 0.71 MTNR1A (0.61) ROCK2MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL6269567 0.71 KCNH2 (0.42) ROCK2KDM4ELMNAHTR1AADRA1D
SCHEMBL2533923 0.70 KCNH2 (0.46) ROCK2KDM4ELMNAHTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337529-A2 HETEROCYCLYLALKYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND COMPOSITIONS CONTAINING SAME Aventis Pharma S.A. (FR) 2003-08-27 EP disclosed
WO-2002040474-A2 HETEROCYCLYLALKYL PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIMICROBIAL AGENTS AVENTIS PHARMA S.A. (FR) 2002-05-23 WO disclosed