SCHEMBL7016833

SCHEMBL7016833

COc1ccc(-c2cc3nnccc3[nH]2)cc1-c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 4/20 0.42
CDK1 P06493 4/20 0.42
CCNB1 P14635 4/20 0.42
GSK3B P49841 4/20 0.42
CDK5 Q00535 4/20 0.42
CDK5R1 Q15078 4/20 0.42
CCNB3 Q8WWL7 4/20 0.42
GSK3A P49840 3/20 0.42
RIPK1 Q13546 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
TP53 P04637 2/20 0.38
HSD17B10 Q99714 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C19 P33261 1/20 0.38
CBFB Q13951 1/20 0.38
NPC1 O15118 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7101502 0.87 CCNB2 (0.44) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL7014990 0.84 RIPK1 (0.48) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL7009747 0.83 CCNB2 (0.63) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL7100815 0.82 RIPK1 (0.42) CCNB2CDK1CCNB1CCNB3RIPK1
SCHEMBL7017680 0.80 RIPK1 (0.43) CCNB2CDK1CCNB1CCNB3RIPK1
SCHEMBL7101268 0.78 RIPK1 (0.43) CCNB2CDK1CCNB1CCNB3RIPK1
SCHEMBL6286415 0.77 TUBB4A (0.38) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL5945897 0.76 ERN1 (0.49) SMN1; SMN2ALDH1A1TP53HSD17B10CYP2D6
SCHEMBL7096737 0.73 NPY5R (0.45) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL6286410 0.73 PARP1 (0.42) KDM4EPOLBJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294718-A2 6,5-FUSED BICYCLIC HETEROCYCLES WARNER-LAMBERT COMPANY LLC (US) 2003-03-26 EP claimed
WO-2001096336-A2 6,5-FUSED BICYCLIC HETEROCYCLES WARNER-LAMBERT COMPANY (US) 2001-12-20 WO claimed