SCHEMBL7101699

SCHEMBL7101699

CC(C)(C)c1ccc2c(c1)OC(C(F)(F)F)CC2C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.35
ALDH1A1 P00352 1/20 0.34
LTB4R Q15722 5/20 0.34
LTB4R2 Q9NPC1 5/20 0.34
FFAR1 O14842 3/20 0.32
PPARG P37231 2/20 0.32
PPARD Q03181 2/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019518 0.78 GRM2 (0.36) ALDH1A1MEN1KMT2A
SCHEMBL7018582 0.73 HCRTR2 (0.36) PTGS1PTGS2PTGDR2MEN1KMT2A
SCHEMBL7103681 0.71 LMNA (0.35) ALDH1A1PPARGPTGS2PTGDR2LMNA
SCHEMBL7103549 0.70 PTPN7 (0.35) ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL7100609 0.70 CYP11B1 (0.31) PTGS2
SCHEMBL7167937 0.70 TSHR (0.42) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL7021904 0.68 CYP1A2 (0.38) ALDH1A1MEN1KMT2ALMNA
SCHEMBL6406400 0.67 LTB4R (0.37) ACHEALDH1A1LTB4RLTB4R2PTGS1
SCHEMBL6405304 0.67 LTB4R (0.37) ACHEALDH1A1LTB4RLTB4R2PTGS1
SCHEMBL9535853 0.66 AKR1B1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1274700-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS Pharmacia Corporation (US) 2003-01-15 EP claimed
WO-2001049675-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS PHARMACIA CORPORATION (US) 2001-07-12 WO claimed
EP-1274700-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS Pharmacia Corporation (US) 2003-01-15 EP disclosed
WO-2001049675-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS PHARMACIA CORPORATION (US) 2001-07-12 WO disclosed