SCHEMBL7101825

SCHEMBL7101825

CCCCCCCCCCC[C@H](CC(=O)C(CCCCCC)C(=O)O)O[Si](C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 9/20 0.42
FFAR1 O14842 2/20 0.42
PPARD Q03181 4/20 0.41
MAPT P10636 1/20 0.41
LCK P06239 1/20 0.41
ZDHHC20 Q5W0Z9 1/20 0.41
ZDHHC2 Q9UIJ5 1/20 0.41
FFAR4 Q5NUL3 1/20 0.39
ACE2 Q9BYF1 1/20 0.39
GRIK1 P39086 1/20 0.36
GRIK2 Q13002 1/20 0.36
PPARG P37231 3/20 0.35
PPARA Q07869 3/20 0.35
TSHR P16473 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
ALDH1A1 P00352 1/20 0.35
SLC22A6 Q4U2R8 1/20 0.35
SLC22A8 Q8TCC7 1/20 0.35
TLR2 O60603 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7108501 0.91 GPR84 (0.39) GPR84FFAR1PPARDMAPTLCK
SCHEMBL7106845 0.87 ZDHHC7 (0.36) GPR84FFAR1MAPTFFAR4TDP1
SCHEMBL27574737 0.87 ZDHHC7 (0.45) GPR84FFAR1FFAR4
SCHEMBL27552552 0.87 ZDHHC7 (0.36) GPR84FFAR1MAPTFFAR4TDP1
SCHEMBL7101909 0.87 ZDHHC7 (0.45) GPR84FFAR1FFAR4
SCHEMBL7103003 0.84 GPR84 (0.53) GPR84FFAR1PPARDMAPTLCK
SCHEMBL7103007 0.84 GPR84 (0.53) GPR84FFAR1PPARDMAPTLCK
SCHEMBL7103210 0.80 ALDH1A1 (0.41) GPR84FFAR1PPARDMAPTLCK
SCHEMBL7103214 0.80 ALDH1A1 (0.41) GPR84FFAR1PPARDMAPTLCK
SCHEMBL28072157 0.79 GPR84 (0.38) GPR84FFAR1PPARDMAPTLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1127886-B1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one HOFFMANN LA ROCHE (CH) 2003-05-07 EP claimed
US-6552204-B1 Lactonization of an acyl halide and a ketene acetal or reacting acyl halide with malonate half acid then cyclizing; high yield ROCHE COLORADO CORPORATION 2003-04-22 US claimed
CN-1319596-A Synthesis of 3,6-dialkyl 5,6-dihydro-4-hydroxide-2H-pyran-2-ketone HOFFMANN LA ROCHE (CH) 2001-10-31 CN claimed
EP-1127886-A1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one F. HOFFMANN-LA ROCHE AG (CH) 2001-08-29 EP claimed
EP-1127886-B1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one HOFFMANN LA ROCHE (CH) 2003-05-07 EP disclosed
EP-1127886-A1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one F. HOFFMANN-LA ROCHE AG (CH) 2001-08-29 EP disclosed