SCHEMBL7103857

SCHEMBL7103857

O=c1[nH]c2ccc(-n3c(=O)c(=O)[nH]c4ccccc43)cc2[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 3/20 0.47
GRIN3B O60391 3/20 0.47
GRIN1 Q05586 3/20 0.47
GRIN2A Q12879 3/20 0.47
GRIN2B Q13224 3/20 0.47
GRIN2C Q14957 3/20 0.47
GRIN3A Q8TCU5 3/20 0.47
KDM4E B2RXH2 3/20 0.47
TSHR P16473 3/20 0.44
PARP1 P09874 1/20 0.42
ALDH1A1 P00352 2/20 0.42
CASP1 P29466 1/20 0.42
OPRM1 P35372 2/20 0.41
OPRD1 P41143 2/20 0.41
OPRK1 P41145 2/20 0.41
OPRL1 P41146 2/20 0.41
TP53 P04637 1/20 0.40
ALOX15 P16050 1/20 0.40
CDC25B P30305 1/20 0.40
GRIA1 P42261 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3150851 0.82 PDE7A (0.51) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL30910102 0.82 PDE7A (0.51) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL26089069 0.79 ADORA3 (0.48) KDM4ETSHRPARP1ALDH1A1CASP1
SCHEMBL30910123 0.79 ADORA3 (0.48) KDM4ETSHRPARP1ALDH1A1CASP1
SCHEMBL23876381 0.72 PARP1 (0.49) KDM4EPARP1ALDH1A1TP53GAA
SCHEMBL5504138 0.71 MAPT (0.45) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL30910121 0.71 OPRM1 (0.48) KDM4EALDH1A1OPRM1OPRL1GAA
SCHEMBL26088643 0.71 OPRM1 (0.48) KDM4EALDH1A1OPRM1OPRL1GAA
SCHEMBL30910120 0.70 OPRM1 (0.50) KDM4ETSHRALDH1A1OPRM1OPRL1
SCHEMBL26092144 0.70 OPRM1 (0.50) KDM4ETSHRALDH1A1OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030207886-A1 Preparation containing quinoxaline derivatives MERCK PATENT GMBH (DE) 2003-11-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030207886-A1 Preparation containing quinoxaline derivatives CUTA, XPA, NQO2 GRIN2D 2658/4885GRIN3B 4215/4885GRIN1 4113/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.