SCHEMBL7112959

SCHEMBL7112959

O=S(=O)(Nc1ncccn1)c1c[c]ccc1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.54
DHFR P00374 1/20 0.54
LMNA P02545 1/20 0.54
TSHR P16473 1/20 0.54
ALDH1A1 P00352 5/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
NPSR1 Q6W5P4 1/20 0.45
KDM4E B2RXH2 3/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
RXFP1 Q9HBX9 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL922001 0.81 AURKA (0.64) AURKADHFRLMNATSHRALDH1A1
SCHEMBL6693457 0.80 LMNA (0.45) LMNAALDH1A1L3MBTL1KMT2ASMN1; SMN2
SCHEMBL332569 0.78 TSHR (0.70) AURKADHFRLMNATSHRALDH1A1
SCHEMBL6312978 0.77 ALDH1A1 (0.57) LMNAALDH1A1KDM4EKMT2AMEN1
SCHEMBL11313543 0.76 CA1 (0.35) LMNATSHRALDH1A1KDM4EKMT2A
SCHEMBL4850048 0.76 KEAP1 (0.66) ALDH1A1KMT2AMEN1MAPTSMN1; SMN2
SCHEMBL6688039 0.73 KMT2A (0.34) AURKADHFRLMNATSHRALDH1A1
SCHEMBL17593233 0.73 ALDH1A1 (0.50) AURKADHFRLMNATSHRALDH1A1
SCHEMBL1043396 0.73 SMN1; SMN2 (0.45) LMNAALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL28435387 0.73 MEN1 (0.38) ALDH1A1KMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140871-A4 THROMBIN OR FACTOR XA INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2004-05-06 EP disclosed
EP-1140871-A1 THROMBIN OR FACTOR XA INHIBITORS Du Pont Pharmaceuticals Company (US) 2001-10-10 EP disclosed
WO-2000039108-A1 THROMBIN OR FACTOR XA INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 2000-07-06 WO disclosed