SCHEMBL711356

SCHEMBL711356

CS(=O)(=O)Nc1cc(NS(=O)(=O)c2ccccc2)cc(C(=O)O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.60
TDP1 Q9NUW8 1/20 0.59
CYTH2 Q99418 1/20 0.55
POLB P06746 1/20 0.55
PFKFB3 Q16875 1/20 0.55
F2 P00734 1/20 0.52
F10 P00742 1/20 0.52
FURIN P09958 1/20 0.52
KEAP1 Q14145 2/20 0.51
IL1RN P18510 1/20 0.51
ERAP1 Q9NZ08 1/20 0.51
CA12 O43570 1/20 0.51
CA9 Q16790 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
AKR1C3 P42330 1/20 0.50
ALDH1A1 P00352 3/20 0.49
PKM P14618 2/20 0.49
GAA P10253 1/20 0.49
ALOX15 P16050 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9818397 0.92 WDR5 (0.69) WDR5TDP1CYTH2POLBPFKFB3
SCHEMBL10487708 0.89 WDR5 (0.73) WDR5TDP1CYTH2POLBPFKFB3
SCHEMBL22653513 0.84 POLB (0.65) POLBPFKFB3CA12CA9MEN1
SCHEMBL29261787 0.83 PFKFB3 (0.68) WDR5TDP1CYTH2POLBPFKFB3
SCHEMBL28538527 0.82 WDR5 (0.73) WDR5TDP1CYTH2POLBPFKFB3
SCHEMBL3447030 0.82 ALDH1A1 (0.53) WDR5TDP1POLBKEAP1MEN1
SCHEMBL894613 0.80 POLB (0.82) POLBPFKFB3KEAP1IL1RNERAP1
SCHEMBL720817 0.78 HPGD (0.58) TDP1KEAP1KMT2AALDH1A1ALOX15
Zinc Ion SCHEMBL9420954 0.78 MEN1 (0.56) WDR5TDP1CYTH2POLBPFKFB3
SCHEMBL9402983 0.78 ALDH1A1 (0.66) WDR5TDP1POLBPFKFB3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8124617-B2 Imidazopyridine compounds TAKEDA SAN DIEGO, INC. (US) 2012-02-28 US disclosed
US-8124617-B2 Imidazopyridine compounds TAKEDA SAN DIEGO, INC. (US) 2012-02-28 US disclosed
US-20100069431-A1 IMIDAZOPYRIDINE COMPOUNDS TAKEDA SAN DIEGO, INC. 2010-03-18 US disclosed
US-20100069431-A1 IMIDAZOPYRIDINE COMPOUNDS TAKEDA SAN DIEGO, INC. 2010-03-18 US disclosed
WO-2007028135-A2 IMIDAZOPYRIDINE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069431-A1 IMIDAZOPYRIDINE COMPOUNDS GCK, GCKR, KHK WDR5 4199/4885TDP1 2189/4885CYTH2 3817/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.