SCHEMBL7115183

SCHEMBL7115183

CCc1ccc(CC)c(C)n1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
NOS3 P29474 1/20 0.34
NOS2 P35228 1/20 0.34
ELANE P08246 2/20 0.34
TKT P29401 1/20 0.34
GRM1 Q13255 1/20 0.31
GABRA1 P14867 2/20 0.31
GABRB2 P47870 2/20 0.31
CTRC Q99895 1/20 0.30
GAA P10253 1/20 0.30
TP53 P04637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17431389 0.85 MEN1 (0.40) PARP1NOS3NOS2TKT
SCHEMBL7150826 0.85 NOS3 (0.37) NOS3NOS2ELANETP53
SCHEMBL21414452 0.78
SCHEMBL10730430 0.78 NOS3 (0.46) PARP1NOS3NOS2ELANETKT
SCHEMBL7573152 0.78 CCR1 (0.40) GRM1
SCHEMBL30585580 0.78 CCR1 (0.40) GRM1
SCHEMBL7118882 0.76 PSMB5 (0.38) PARP1NOS3NOS2ELANETKT
SCHEMBL25907277 0.76 ALDH1A1 (0.37) PARP1NOS3NOS2ELANEGAA
SCHEMBL19242233 0.75 ELANE (0.36) PARP1ELANEGABRA1GABRB2CTRC
SCHEMBL21604163 0.74 NOS3 (0.42) PARP1NOS3NOS2TKTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106854207-A Dai piperazine analog derivative, its preparation method, pharmaceutical composition and purposes 上海赛默罗生物科技有限公司 2017-06-16 CN disclosed
US-20030064989-A1 Inhibitors of cell proliferation, angiogenesis, fertility, and muscle contraction REGENTS OF THE UNIVERSITY OF CALIFORNIA, THE 2003-04-03 US disclosed
US-4871848-A OIL, GAS WELLS CORROSION INHIBITORS THE DOW CHEMICAL COMPANY (US) 1989-10-03 US disclosed
US-4740320-A REACTION OF NITROGEN-CONTAINING AROMATIC HETEROCYCLIC COMPONENT, KETONE OR ALDEHYDE, AMINE OR POLYAMINE THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed
US-4725373-A CORROSION RESISTANCE FOR METAL TOOLS AND EQUIPMENT USED IN OIL AND GAS WELLS THE DOW CHEMICAL COMPANY (US) 1988-02-16 US disclosed
US-4724003-A Asphalt compositions containing anti-stripping additives prepared from hydrocarbyl substituted nitrogen-containing aromatic heterocyclic compounds, aldehydes or ketones and amines THE DOW CHEMICAL COMPANY (US) 1988-02-09 US disclosed
US-4676834-A Novel compositions prepared from methyl substituted nitrogen-containing aromatic heterocyclic compounds and an aldehyde or ketone THE DOW CHEMICAL COMPANY (US) 1987-06-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030064989-A1 Inhibitors of cell proliferation, angiogenesis, fertility, and muscle contraction MYH10, MYLK, MKI67 PARP1 866/4885NOS3 416/4885NOS2 1820/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.