SCHEMBL7115993

SCHEMBL7115993

CCC(=O)Oc1cc(Br)c(Oc2ccc(OC)cc2)c(Br)c1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.39
KMT2A Q03164 6/20 0.38
ESR1 P03372 2/20 0.38
HIF1A Q16665 2/20 0.38
RECQL P46063 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 3/20 0.38
ATM Q13315 1/20 0.38
GAA P10253 4/20 0.37
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
ACHE P22303 2/20 0.36
MEN1 O00255 3/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7116011 0.86 THRA (0.40) L3MBTL1KMT2AESR1HIF1ARECQL
SCHEMBL5282022 0.86 BACE1 (0.48) KMT2ASMN1; SMN2GAATHRATHRB
SCHEMBL7119529 0.83 KMT2A (0.45) L3MBTL1KMT2AESR1HIF1ARECQL
SCHEMBL7116646 0.82 THRB (0.44) L3MBTL1KMT2AHIF1ASMN1; SMN2THRA
SCHEMBL5277949 0.75 THRA (0.43) KMT2ATHRATHRBCYP3A4MEN1
SCHEMBL7122561 0.74 ACHE (0.41) KMT2AESR1HIF1ARECQLSMN1; SMN2
SCHEMBL9037509 0.74 ESR1 (0.45) KMT2AESR1HIF1ARECQLSMN1; SMN2
SCHEMBL5283822 0.73 THRB (0.57) THRATHRB
SCHEMBL5283377 0.71 THRA (0.37) THRATHRBCYP3A4HTTKDM4E
SCHEMBL6156093 0.71 THRB (0.54) THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358175-A2 PHENOXY SUBSTITUTED BENZOCONDENSED HETEROARYL DERIVATIVES AS THYROID RECEPTOR LIGANDS KARO BIO AB (SE) 2003-11-05 EP disclosed
WO-2002062780-A2 PHENOXY SUBSTITUTED BENZOCONDENSED HETEROARYL DERIVATIVES AS THYROID RECEPTOR LIGANDS KARO BIO AB (SE) 2002-08-15 WO disclosed