SCHEMBL7115995

SCHEMBL7115995

COC(=O)C(C)c1cc(Br)c(Oc2ccc(OC)cc2)c(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RAB9A P51151 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPBWR1 P48145 1/20 0.40
MCHR1 Q99705 1/20 0.40
PTGS2 P35354 4/20 0.40
PTGS1 P23219 3/20 0.40
ALDH1A1 P00352 1/20 0.39
AKR1C3 P42330 2/20 0.39
AKR1C2 P52895 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5858288 0.87 PTGS2 (0.54) THRATHRBCYP1A2CYP2C19NPBWR1
SCHEMBL7050847 0.83 THRB (0.54) THRATHRB
SCHEMBL7116014 0.83 THRA (0.40) MEN1KMT2AMAPTTHRATHRB
SCHEMBL7116655 0.82 THRB (0.47) MEN1KMT2ATHRATHRBCYP1A2
SCHEMBL4007061 0.78 MEN1 (0.54) TDP1L3MBTL1RAB9AMEN1KMT2A
SCHEMBL8745429 0.76 THRB (0.48) THRATHRBPTGS2ALDH1A1TSHR
SCHEMBL5964846 0.75 THRA (0.48) THRATHRBCYP1A2PTGS2PTGS1
SCHEMBL7050577 0.75 FOLH1 (0.50) TDP1KMT2ACYP3A4PTGS2PTGS1
SCHEMBL7112160 0.74 BACE1 (0.52) RAB9AMEN1KMT2ANPC1MAPT
SCHEMBL3925861 0.74 THRA (0.37) MAPTTHRATHRBNPBWR1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358175-A2 PHENOXY SUBSTITUTED BENZOCONDENSED HETEROARYL DERIVATIVES AS THYROID RECEPTOR LIGANDS KARO BIO AB (SE) 2003-11-05 EP disclosed
WO-2002062780-A2 PHENOXY SUBSTITUTED BENZOCONDENSED HETEROARYL DERIVATIVES AS THYROID RECEPTOR LIGANDS KARO BIO AB (SE) 2002-08-15 WO disclosed