SCHEMBL7119688

SCHEMBL7119688

CCOC(=O)c1cn(CC)c2cc(OS(=O)(=O)C(F)(F)F)c(F)cc2c1=O

nearest known ligand 0.71

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 7/20 0.57
ALDH1A1 P00352 6/20 0.57
KDM4E B2RXH2 5/20 0.57
HSD17B10 Q99714 5/20 0.57
KMT2A Q03164 3/20 0.56
LMNA P02545 3/20 0.53
POLB P06746 2/20 0.51
MEN1 O00255 2/20 0.48
MAPT P10636 1/20 0.48
THRB P10828 1/20 0.48
NPC1 O15118 1/20 0.46
DRD3 P35462 1/20 0.45
HTT P42858 2/20 0.44
BRD4 O60885 1/20 0.44
TSHR P16473 1/20 0.44
CYP2J2 P51589 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10412669 0.91 ALDH1A1 (0.48) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL4296349 0.85 ADRB2 (0.47) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL7128071 0.83 KMT2A (0.76) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL10413494 0.83 ALDH1A1 (0.45) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL10412625 0.81 KMT2A (0.48) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL10824134 0.81 HSD17B10 (0.63) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL8041564 0.79 POLB (0.69) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL6687806 0.79 LMNA (0.67) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL29823822 0.79 POLB (0.69) HPGDALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL10575415 0.79 KMT2A (0.67) HPGDALDH1A1KDM4EHSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed
US-4945160-A Preparation of certain 7-substituted quinolones WARNER-LAMBERT COMPANY (US) 1990-07-31 US disclosed