SCHEMBL7121914

SCHEMBL7121914

CN(C)CC(=O)NC1SC=C(N(CC(=O)O)C(=O)c2ccccc2)N1CN.NC(=O)c1ccc2c(c1)CCC2

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.35
NOD2 Q9HC29 1/20 0.33
NOD1 Q9Y239 1/20 0.33
MAPK14 Q16539 2/20 0.32
TRPC6 Q9Y210 1/20 0.31
HSD17B3 P37058 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
MEN1 O00255 1/20 0.30
HPGD P15428 1/20 0.30
RAD52 P43351 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7129076 0.92 SMYD3 (0.35) SMYD3NOD2NOD1MAPK14SMN1; SMN2
SCHEMBL7129797 0.87 MAPK14 (0.32) SMYD3NOD2NOD1MAPK14HSD17B3
Trifluoroacetic Acid SCHEMBL7426138 0.79 OPRM1 (0.35)
Trifluoroacetic Acid SCHEMBL7128334 0.79 OPRM1 (0.34)
Trifluoroacetic Acid SCHEMBL7129463 0.70 ACHE (0.35)
SCHEMBL7121817 0.70 HSD17B3 (0.41) HSD17B3
SCHEMBL7131862 0.68 RXRA (0.36) SMYD3MAPK14HSD17B3SMN1; SMN2ALDH1A1
SCHEMBL4805867 0.68 MAPT (0.38) SMYD3NOD2NOD1MAPK14TRPC6
Hydrochloric Acid SCHEMBL7128388 0.68 RXRA (0.36) MAPK14HSD17B3SMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL7427799 0.68 MAPK14 (0.36) SMYD3MAPK14HSD17B3SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294691-A1 SERINE PROTEASE INHIBITORS Tularik Limited (GB) 2003-03-26 EP disclosed
WO-2001096305-A1 SERINE PROTEASE INHIBITORS TULARIK LIMITED (GB) 2001-12-20 WO disclosed