SCHEMBL7121817

SCHEMBL7121817

CC(=O)N1CCC(N(CC(=O)O)C(=O)c2ccccc2)CC1.NC(=O)c1ccc2c(c1)CCC2

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 1/20 0.41
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
OPRK1 P41145 2/20 0.39
CHRM2 P08172 1/20 0.39
CHRM3 P20309 1/20 0.39
MCHR1 Q99705 4/20 0.38
UBE2M P61081 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
F10 P00742 2/20 0.36
ENPP2 Q13822 1/20 0.36
LIMK2 P53671 1/20 0.36
KDM5A P29375 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4803612 0.86 TPSAB1 (0.41) OPRM1OPRD1OPRK1F10
SCHEMBL4813549 0.81 SMYD3 (0.38) OPRM1OPRD1OPRK1CHRM2CHRM3
Trifluoroacetic Acid SCHEMBL4810746 0.78 F2 (0.38) OPRM1OPRD1OPRK1UBE2MDCUN1D1
SCHEMBL4812628 0.77 GPR119 (0.42)
SCHEMBL4810407 0.76 OPRM1 (0.42) HSD17B3OPRM1OPRD1OPRK1MCHR1
Trifluoroacetic Acid SCHEMBL7434362 0.76 OPRM1 (0.37) OPRM1OPRD1F10
Trifluoroacetic Acid SCHEMBL4807393 0.73 AGER (0.39)
Trifluoroacetic Acid SCHEMBL4810923 0.71 DCUN1D1 (0.36) OPRM1OPRD1DCUN1D1F10
Trifluoroacetic Acid SCHEMBL7433732 0.70 SLC6A2 (0.34) OPRM1OPRD1
SCHEMBL7121914 0.70 SMYD3 (0.35) HSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294691-A1 SERINE PROTEASE INHIBITORS Tularik Limited (GB) 2003-03-26 EP disclosed
EP-1240154-A1 SERINE PROTEASE INHIBITORS Tularik Limited (GB) 2002-09-18 EP disclosed
WO-2001096305-A1 SERINE PROTEASE INHIBITORS TULARIK LIMITED (GB) 2001-12-20 WO disclosed
WO-2001044226-A1 SERINE PROTEASE INHIBITORS TULARIK LIMITED (GB) 2001-06-21 WO disclosed