SCHEMBL7123604

SCHEMBL7123604

O=C(O)CN(c1ccc(Br)cc1)S(=O)(=O)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 6/20 0.46
NFE2L2 Q16236 6/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.41
PPARG P37231 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
NR1I2 O75469 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14855516 0.82 L3MBTL1 (0.47) KEAP1NFE2L2L3MBTL1SMN1; SMN2HTT
SCHEMBL7117168 0.79 NR1I2 (0.40) L3MBTL1TSHRHTTNR1I2
SCHEMBL1409649 0.79 SMN1; SMN2 (0.63) KEAP1NFE2L2L3MBTL1SMN1; SMN2TSHR
SCHEMBL7118481 0.75 MCL1 (0.44) L3MBTL1TSHRHTTNR1I2
SCHEMBL7922299 0.72 L3MBTL1 (0.45) L3MBTL1SMN1; SMN2TSHRNR1I2
SCHEMBL3366459 0.72 KEAP1 (0.86) KEAP1NFE2L2PPARGTSHR
SCHEMBL7119808 0.71 KIF11 (0.42) L3MBTL1TSHRHTT
SCHEMBL340532 0.70 MEN1 (0.42) KEAP1NFE2L2L3MBTL1
SCHEMBL8818175 0.69 CA2 (0.40)
SCHEMBL7119429 0.69 CNR2 (0.46) L3MBTL1SMN1; SMN2TSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed