SCHEMBL7125002

SCHEMBL7125002

CNC(=O)c1ccccc1OCCN(CCCCNC(=O)c1ccccc1)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.49
SIGMAR1 Q99720 7/20 0.47
TMEM97 Q5BJF2 6/20 0.47
ALDH1A1 P00352 1/20 0.47
HCRTR1 O43613 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HIF1A Q16665 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ACKR3 P25106 1/20 0.46
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7129202 0.87 NPC1 (0.53) APPSIGMAR1TMEM97ACKR3DRD2
SCHEMBL7126384 0.81 SIGMAR1 (0.47) APPSIGMAR1TMEM97ALDH1A1ACKR3
SCHEMBL8063854 0.81 KDM4E (0.51) APPSIGMAR1TMEM97ALDH1A1MEN1
SCHEMBL7573340 0.80 POLB (0.50) SIGMAR1TMEM97ALDH1A1MEN1KMT2A
SCHEMBL7129442 0.77 SIGMAR1 (0.60) APPSIGMAR1TMEM97ACKR3DRD2
SCHEMBL7169601 0.77 SIGMAR1 (0.57) APPSIGMAR1TMEM97ACKR3DRD2
SCHEMBL13579952 0.72 SIGMAR1 (0.83) APPSIGMAR1TMEM97ACKR3
SCHEMBL4753614 0.71 ALDH1A1 (0.54) ALDH1A1HCRTR1MEN1KMT2ADRD2
SCHEMBL30576437 0.70 APP (0.59) APPSIGMAR1TMEM97ACKR3
SCHEMBL10621481 0.70 TMEM97 (0.59) SIGMAR1TMEM97ACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6670400-B1 Secretion inhibitors for gastric acid, antiemetics; N(4-(2-(2-methoxyphenoxy)ethyl)aminobutyl)benzamide; SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2003-12-30 US disclosed
EP-0820434-B1 PHENOXYETHYLAMINE DERIVATIVES HAVING HIGH AFFINITY FOR THE 5-HT 1A RECEPTOR, PREPARATION THEREOF, USE THEREOF AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES SOD CONSEILS RECH APPLIC (FR) 2000-08-09 EP disclosed