SCHEMBL7127715

SCHEMBL7127715

COC(=O)c1c(C2C=CCC2)cc2c(c1-c1ccc(F)cc1)C(=O)CC(C)(C)C2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.34
ALDH1A1 P00352 5/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 2/20 0.34
GCGR P47871 1/20 0.34
LMNA P02545 3/20 0.33
BUB1 O43683 1/20 0.32
SLC6A3 Q01959 4/20 0.32
SLC6A4 P31645 3/20 0.32
OPRM1 P35372 1/20 0.31
GFER P55789 1/20 0.31
NPSR1 Q6W5P4 2/20 0.30
HTT P42858 1/20 0.30
SSTR5 P35346 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6421909 0.85 MAPT (0.33) ALPLMAPTBUB1
SCHEMBL7123071 0.85 ALPL (0.36) ALPLALDH1A1MEN1KMT2ACYP1A2
SCHEMBL7122832 0.80 ALPL (0.40) ALPLALDH1A1MEN1KMT2ACYP1A2
SCHEMBL6376468 0.77 GCGR (0.38) ALPLALDH1A1MEN1KMT2ACYP1A2
SCHEMBL6422071 0.72 ALPL (0.35) ALPLALDH1A1MAPTBUB1SLC6A3
SCHEMBL18863342 0.69 SLC6A4 (0.38) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL6484099 0.69 CYP1A2 (0.48) ALPLALDH1A1MEN1KMT2ACYP1A2
SCHEMBL6422907 0.68 ALPL (0.39) ALPLALDH1A1MEN1KMT2ACYP1A2
SCHEMBL6423040 0.62 ALPL (0.34) ALPLMEN1KMT2AMAPTBUB1
SCHEMBL22952259 0.60 KDM4E (0.47) ALDH1A1MAPTLMNASLC6A3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6586613-B1 Compounds such as 5-(tert-butyldimethylsiloxy)-7,7-dimethyl -4(4-fluorophenyl)-3-(hydroxy-(4-trifluorophenyl)-methyl)-2-isopropyl -5,6,7,8-tetrahydronaphthalene, used as antagonists for cholesteryl ester transferase protein; hyperlipemia BAYER AKTIENGELLSCHAFT (DE) 2003-07-01 US disclosed