SCHEMBL7123071

SCHEMBL7123071

COC(=O)c1c(C2CCCC2)cc2c(c1-c1ccc(F)cc1)C(=O)CC(C)(C)C2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.36
PTGDR Q13258 1/20 0.36
ALDH1A1 P00352 5/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP3A4 P08684 1/20 0.36
SLC6A3 Q01959 3/20 0.36
SLC6A4 P31645 2/20 0.36
MAPT P10636 2/20 0.36
OPRM1 P35372 1/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 2/20 0.34
TSHR P16473 1/20 0.34
GCGR P47871 1/20 0.34
TP53 P04637 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7127715 0.85 ALPL (0.34) ALPLALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6422071 0.84 ALPL (0.35) ALPLPTGDR2PTGDRALDH1A1SLC6A3
SCHEMBL7122832 0.83 ALPL (0.40) ALPLALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6484099 0.79 CYP1A2 (0.48) ALPLALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6376468 0.78 GCGR (0.38) ALPLALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6421909 0.72 MAPT (0.33) ALPLMAPTBUB1
SCHEMBL6422907 0.71 ALPL (0.39) ALPLALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7128683 0.71 CETP (0.43) PTGDR2PTGDR
SCHEMBL6421617 0.69 CETP (0.42) PTGDR2PTGDRSLC6A3SLC6A4
SCHEMBL8129664 0.68 MAPT (0.45) ALPLALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6586613-B1 Compounds such as 5-(tert-butyldimethylsiloxy)-7,7-dimethyl -4(4-fluorophenyl)-3-(hydroxy-(4-trifluorophenyl)-methyl)-2-isopropyl -5,6,7,8-tetrahydronaphthalene, used as antagonists for cholesteryl ester transferase protein; hyperlipemia BAYER AKTIENGELLSCHAFT (DE) 2003-07-01 US disclosed