SCHEMBL7128554

SCHEMBL7128554

NC(=O)c1ccc(-c2ccncc2)o1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.64
HPGD P15428 2/20 0.64
KDM4E B2RXH2 2/20 0.64
LMNA P02545 1/20 0.64
PRNP P04156 1/20 0.64
HSD17B10 Q99714 1/20 0.64
SLC9A1 P19634 3/20 0.46
CYP17A1 P05093 1/20 0.45
CDC7 O00311 2/20 0.43
DBF4 Q9UBU7 2/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
PDE4B Q07343 2/20 0.42
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
CHUK O15111 1/20 0.41
POLB P06746 1/20 0.41
HSD17B1 P14061 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27605036 0.85 ALDH1A1 (0.47) ALDH1A1HPGDKDM4ELMNAPRNP
SCHEMBL5735008 0.83 ALDH1A1 (0.65) ALDH1A1HPGDKDM4EPDE4B
Hydrochloric Acid SCHEMBL5542925 0.81 ALDH1A1 (0.62) ALDH1A1HPGDKDM4EPDE4B
SCHEMBL14395763 0.81 ALDH1A1 (0.44) ALDH1A1HPGDKDM4ELMNAPRNP
SCHEMBL4252554 0.81 ALDH1A1 (0.44) ALDH1A1HPGDKDM4ELMNAPRNP
SCHEMBL4163540 0.81 ALDH1A1 (0.68) ALDH1A1HPGDKDM4ELMNAPRNP
SCHEMBL3420262 0.80 CYP2A6 (0.54) ALDH1A1HPGDKDM4ELMNAPRNP
SCHEMBL2031645 0.79 ALDH1A1 (0.71) ALDH1A1HPGDKDM4ELMNAPRNP
SCHEMBL5735703 0.79 ABL1 (0.52) ALDH1A1HPGDKDM4EHSD17B10HSD17B1
SCHEMBL12885825 0.78 ALDH1A1 (0.69) ALDH1A1HPGDKDM4ELMNAPRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100345847-C Novel biarylcarboxamides ASTRAZENECA AB (SE) 2007-10-31 CN claimed
CN-1400973-A Novel biarylcarboxamides ASTRAZENECA AB (SE) 2003-03-05 CN claimed
EP-4646263-A1 SPRK1 INHIBITORS AND METHODS OF USE Allianthera (Suzhou) Biopharmaceutical Co., Ltd. (CN) 2025-11-12 EP disclosed
US-12325704-B2 SRPK1 inhibitors EXONATE LIMITED (GB) 2025-06-10 US disclosed
WO-2024155864-A1 SPRK1 INHIBITORS AND METHODS OF USE ALLIANTHERA (SUZHOU) BIOPHARMACEUTICAL CO., LTD. (CN) 2024-07-25 WO disclosed
CN-111448193-B SRPK1 inhibitors 埃克森纳特有限公司 2023-12-22 CN disclosed
CN-108738319-B Compounds for anti-angiogenic therapy or prophylaxis 埃克森纳特有限公司 2023-09-29 CN disclosed
US-20220389015-A1 SRPK1 INHIBITORS EXONATE LIMITED (GB) 2022-12-08 US disclosed
US-11420969-B2 SRPK1 inhibitors EXONATE LIMITED (GB) 2022-08-23 US disclosed
CN-100345847-C Novel biarylcarboxamides ASTRAZENECA AB (SE) 2007-10-31 CN disclosed
CN-1400973-A Novel biarylcarboxamides ASTRAZENECA AB (SE) 2003-03-05 CN disclosed
US-20030008867-A1 Compounds ASTRAZENECA AB (SE) 2003-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030008867-A1 Compounds DRD2, DRD1, GRIN2A ALDH1A1 75/4885HPGD 1662/4885KDM4E 2318/4885
US-11420969-B2 SRPK1 inhibitors SRPK1, SRPK3, SRPK2 ALDH1A1 4429/4885HPGD 3277/4885KDM4E 3360/4885
US-20220389015-A1 SRPK1 INHIBITORS SRPK1, SRPK3, SRPK2 ALDH1A1 4429/4885HPGD 3277/4885KDM4E 3360/4885
US-12325704-B2 SRPK1 inhibitors SRPK1, SRPK3, SRPK2 ALDH1A1 4429/4885HPGD 3277/4885KDM4E 3360/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.