SCHEMBL7142883

SCHEMBL7142883

Cc1cc(C)cc(S(=O)(=O)c2ccc([N+](=O)[O-])cc2)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.55
TSHR P16473 2/20 0.55
HSD17B10 Q99714 1/20 0.55
KMT2A Q03164 3/20 0.53
POLB P06746 1/20 0.53
HSP90AA1 P07900 1/20 0.51
CXCR5 P32302 1/20 0.51
APLNR P35414 1/20 0.51
RAB9A P51151 1/20 0.51
CCR6 P51684 1/20 0.51
GFER P55789 1/20 0.51
CA1 P00915 5/20 0.50
CA2 P00918 5/20 0.50
CA12 O43570 4/20 0.50
CA9 Q16790 4/20 0.50
CA14 Q9ULX7 4/20 0.50
CA3 P07451 3/20 0.50
CA4 P22748 3/20 0.50
CA6 P23280 3/20 0.50
CA5A P35218 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6577803 0.86 ACHE (0.75) ACHEHSD17B10KMT2APOLBHSP90AA1
SCHEMBL8866076 0.84 KMT2A (0.64) ACHETSHRHSD17B10KMT2APOLB
SCHEMBL12550497 0.84 GAA (0.67) TSHRKMT2APOLBCA2GAA
SCHEMBL11419996 0.84 CA2 (0.67) ACHEHSD17B10KMT2APOLBCA1
SCHEMBL3158508 0.84 CA2 (0.67) ACHEHSD17B10KMT2APOLBCA1
SCHEMBL11855965 0.84 CA2 (0.67) ACHEHSD17B10KMT2APOLBCA1
Sulfuric Acid SCHEMBL28487498 0.81 ACHE (0.67) ACHEHSD17B10KMT2APOLBHSP90AA1
SCHEMBL12409036 0.80 GAA (0.76) TSHRKMT2AHSP90AA1CA1CA2
SCHEMBL2762326 0.79 ALDH1A1 (0.75) TSHRKMT2APOLBCA1CA2
SCHEMBL11854911 0.78 CA1 (0.70) KMT2APOLBCA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0930302-B1 Benzosulfone derivatives HOFFMANN LA ROCHE (CH) 2003-04-02 EP disclosed
US-5990105-A POSSESS A SELECTIVE AFFINITY TO 5HT-6 RECEPTORS; TREATING OR PREVENTING PSYCHOSES, SCHIZOPHRENIA, MANIC DEPRESSIONS, DEPRESSIONS, NEUROLOGICAL DISORDERS, PARKINSON'S, AMYOTROPHIC LATERAL SCLEROSIS, ALZHEIMER'S AND HUNTINGTON'S DISEASE HOFFMANN-LA ROCHE INC. (US) 1999-11-23 US disclosed
EP-0930302-A2 Benzosulfone derivatives F.HOFFMANN-LA ROCHE AG (CH) 1999-07-21 EP disclosed