SCHEMBL7143142

SCHEMBL7143142

COc1ccc(-c2ccccc2C)n2nc(N)nc12

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.48
PDE10A Q9Y233 3/20 0.46
NUDT1 P36639 2/20 0.46
PDE4D Q08499 5/20 0.46
HSP90AB1 P08238 5/20 0.41
MAPT P10636 4/20 0.40
THRB P10828 1/20 0.40
HSP90AA1 P07900 2/20 0.39
PDE2A O00408 1/20 0.38
PDE6D O43924 1/20 0.38
PDE6A P16499 1/20 0.38
PDE6G P18545 1/20 0.38
PDE4A P27815 1/20 0.38
PDE6B P35913 1/20 0.38
PDE6C P51160 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE6H Q13956 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7045163 0.85 JAK2 (0.47) JAK2PDE10ANUDT1PDE4DHSP90AB1
SCHEMBL7148123 0.85 NUDT1 (0.55) JAK2PDE10ANUDT1PDE4DHSP90AB1
SCHEMBL2250839 0.82 PDE4D (0.64) JAK2PDE10ANUDT1PDE4DHSP90AB1
SCHEMBL7144538 0.78 PDE4D (0.49) PDE10APDE4DHSP90AB1MAPT
SCHEMBL7145674 0.76 PDE10A (0.50) PDE10APDE4DHSP90AB1
SCHEMBL7043078 0.75 JAK1 (0.60) PDE10APDE4DHSP90AB1MAPT
SCHEMBL2257907 0.74 MAPT (0.49) JAK2PDE10APDE4DHSP90AB1MAPT
SCHEMBL7146898 0.74 KDM4E (0.51) PDE10APDE4D
SCHEMBL7043841 0.74 MAPT (0.51) PDE10APDE4DHSP90AB1MAPT
SCHEMBL4066707 0.73 PDE10A (0.45) JAK2PDE10APDE4DHSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514989-B1 Has a good affinity to the adenosine receptor and can therefore be used for the treatment or protection of diseases mediated by this receptor HOFFMANN-LA ROCHE INC. 2003-02-04 US disclosed