SCHEMBL7143457

SCHEMBL7143457

CCCCCCc1ccc(C(=O)C(Br)c2ccncc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
THRA P10827 8/20 0.50
THRB P10828 8/20 0.50
RARB P10826 5/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 1/20 0.49
RARA P10276 1/20 0.49
MAPT P10636 1/20 0.49
MTOR P42345 1/20 0.49
TRPV1 Q8NER1 3/20 0.47
PLA2G1B P04054 1/20 0.46
ATG4B Q9Y4P1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6276185 0.99 THRA (0.49) THRATHRBRARBMEN1KMT2A
SCHEMBL7148129 0.95 RARB (0.47) THRATHRBRARBALDH1A1MAPT
Bromide SCHEMBL6282038 0.93 RARB (0.46) THRATHRBRARBALDH1A1MAPT
SCHEMBL7140352 0.89 KMT2A (0.46) THRBMEN1KMT2AALDH1A1MAPT
Bromide SCHEMBL6285577 0.88 KMT2A (0.45) THRBMEN1KMT2AALDH1A1MAPT
SCHEMBL7142545 0.83 RAB9A (0.46) KMT2AALDH1A1MAPTTRPV1
SCHEMBL7139170 0.77 RARB (0.57) THRATHRBRARBMEN1KMT2A
SCHEMBL7147231 0.75 ALDH1A1 (0.42) KMT2AALDH1A1
SCHEMBL9667265 0.75 THRA (0.61) THRATHRBRARBMEN1KMT2A
SCHEMBL9667141 0.75 THRA (0.61) THRATHRBRARBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed