SCHEMBL7148129

SCHEMBL7148129

CCCCc1ccc(C(=O)C(Br)c2ccncc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 3/20 0.47
PLK1 P53350 1/20 0.47
THRA P10827 3/20 0.46
THRB P10828 3/20 0.46
TRPV1 Q8NER1 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
NFKB1 P19838 1/20 0.42
S1PR1 P21453 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6282038 0.99 RARB (0.46) RARBPLK1THRATHRBTRPV1
SCHEMBL7143457 0.95 THRA (0.50) RARBTHRATHRBTRPV1ALDH1A1
Bromide SCHEMBL6276185 0.93 THRA (0.49) RARBTHRATHRBTRPV1ALDH1A1
SCHEMBL7140352 0.92 KMT2A (0.46) PLK1THRBTRPV1SMN1; SMN2LMNA
Bromide SCHEMBL6285577 0.90 KMT2A (0.45) PLK1THRBTRPV1SMN1; SMN2LMNA
SCHEMBL7142545 0.85 RAB9A (0.46) PLK1TRPV1SMN1; SMN2LMNAHTT
Bromide SCHEMBL6284151 0.84 RAB9A (0.45) PLK1TRPV1SMN1; SMN2LMNAHTT
SCHEMBL7147231 0.77 ALDH1A1 (0.42) SMN1; SMN2LMNAHTTALDH1A1HPGD
SCHEMBL9641063 0.77 RARB (0.56) RARBPLK1THRATHRBTRPV1
Bromide SCHEMBL6282584 0.76 ALDH1A1 (0.41) SMN1; SMN2LMNAHTTALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed