SCHEMBL7144741

SCHEMBL7144741

CC(C)(C)c1ccc(C(=O)C(Br)c2ccncc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KIF11 P52732 1/20 0.44
GSK3B P49841 1/20 0.44
KIT P10721 1/20 0.42
SRC P12931 1/20 0.42
FLT3 P36888 1/20 0.42
ITK Q08881 1/20 0.42
HDAC1 Q13547 1/20 0.42
MAPT P10636 4/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
TP53 P04637 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SRD5A2 P31213 1/20 0.41
LMNA P02545 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6280874 0.98 ALDH1A1 (0.43) ALDH1A1TSHRHSD17B10KIF11GSK3B
SCHEMBL6619666 0.94 ALDH1A1 (0.44) ALDH1A1TSHRHSD17B10KIF11GSK3B
Bromide SCHEMBL6545831 0.92 ALDH1A1 (0.43) ALDH1A1TSHRHSD17B10KIF11GSK3B
Bromide SCHEMBL6600773 0.87 MAPT (0.39) ALDH1A1TSHRHSD17B10KIF11GSK3B
SCHEMBL7149547 0.86 GSK3B (0.62) KIF11GSK3BSRD5A2NAMPTHIF1A
Bromide SCHEMBL6284163 0.84 GSK3B (0.60) KIF11GSK3BSRD5A2NAMPTHIF1A
SCHEMBL7143608 0.82 RAB9A (0.53) ALDH1A1KIF11MAPTNPC1RAB9A
SCHEMBL7147231 0.82 ALDH1A1 (0.42) ALDH1A1GSK3BITKNPC1RAB9A
Bromide SCHEMBL6282388 0.81 RAB9A (0.52) ALDH1A1KIF11MAPTNPC1RAB9A
SCHEMBL21990365 0.81 ALDH1A1 (0.48) ALDH1A1TSHRHSD17B10GSK3BHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed