SCHEMBL7143608

SCHEMBL7143608

CC(C)(C)c1ccc(C(=O)C(Br)c2cccnc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.53
NPC1 O15118 2/20 0.53
NAMPT P43490 3/20 0.51
ALDH1A1 P00352 3/20 0.50
MAPT P10636 3/20 0.50
LMNA P02545 2/20 0.50
HTT P42858 1/20 0.50
THRB P10828 2/20 0.49
KIF11 P52732 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
ALOX12 P18054 1/20 0.44
TP53 P04637 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6282388 0.99 RAB9A (0.52) RAB9ANPC1NAMPTALDH1A1MAPT
SCHEMBL7142799 0.84 NAMPT (0.49) RAB9ANPC1NAMPTALDH1A1MAPT
Bromide SCHEMBL6276160 0.83 NAMPT (0.48) RAB9ANPC1NAMPTALDH1A1MAPT
SCHEMBL7144741 0.82 ALDH1A1 (0.44) RAB9ANPC1NAMPTALDH1A1MAPT
SCHEMBL7149156 0.82 CYP17A1 (0.49) RAB9AALDH1A1MAPTLMNAHTT
SCHEMBL7140967 0.82 SMN1; SMN2 (0.51) NAMPTALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL7144713 0.81 CYP19A1 (0.53) RAB9ANPC1NAMPTALDH1A1MAPT
SCHEMBL7149214 0.81 POLB (0.51) RAB9AALDH1A1LMNATHRBSMN1; SMN2
Bromide SCHEMBL6279795 0.81 CYP17A1 (0.48) RAB9ANPC1ALDH1A1MAPTLMNA
Bromide SCHEMBL6280874 0.81 ALDH1A1 (0.43) RAB9ANPC1NAMPTALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed