SCHEMBL7147314

SCHEMBL7147314

Cc1nc2sccn2c(=O)c1CCN1CCC(n2ccc3ccccc32)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.54
MAPT P10636 3/20 0.54
TSHR P16473 3/20 0.54
TDP1 Q9NUW8 3/20 0.54
ALDH1A1 P00352 2/20 0.54
LMNA P02545 2/20 0.54
TP53 P04637 2/20 0.54
CYP2C9 P11712 2/20 0.54
ALOX15 P16050 2/20 0.54
DGKA P23743 2/20 0.54
HSD17B10 Q99714 2/20 0.54
KDM4E B2RXH2 2/20 0.54
CYP2C19 P33261 1/20 0.54
DRD2 P14416 7/20 0.53
HTR1A P08908 7/20 0.53
HTR2A P28223 7/20 0.53
ADRA1A P35348 4/20 0.53
HTR2C P28335 3/20 0.53
ADRA2A P08913 3/20 0.53
ADRA2B P18089 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7142123 0.88 HTR2A (0.59) CYP2D6MAPTTSHRTDP1ALDH1A1
SCHEMBL7150338 0.84 DRD2 (0.51) CYP2D6MAPTTSHRTDP1ALDH1A1
SCHEMBL7149529 0.84 DRD2 (0.53) CYP2D6MAPTTSHRTDP1ALDH1A1
SCHEMBL6617444 0.80 ALDH1A1 (0.55) CYP2D6MAPTTSHRTDP1ALDH1A1
SCHEMBL7145335 0.80 DRD2 (0.52) CYP2D6MAPTTSHRCYP2C9KDM4E
SCHEMBL7699102 0.77 DRD2 (0.54) CYP2D6MAPTTSHRTDP1ALDH1A1
SCHEMBL12786167 0.76 ALDH1A1 (0.56) CYP2D6MAPTTSHRTDP1ALDH1A1
SCHEMBL10944718 0.75 ALDH1A1 (0.51) CYP2D6MAPTTSHRTDP1ALDH1A1
SCHEMBL10922663 0.75 CYP2D6 (0.51) CYP2D6MAPTTSHRTDP1ALDH1A1
SCHEMBL15999621 0.74 HTR1A (0.65) CYP2D6MAPTTSHRTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808313-B1 ANTIPSYCHOTIC 4-(1H-INDOLYL-1-YL)-1-SUBSTITUTED PIPERIDINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2003-08-13 EP disclosed