Water

Water

SCHEMBL714855

O.O=C(O)c1ccc(C(=O)O)c2c(C(=O)O)ccc(C(=O)O)c12

nearest known ligand 0.93

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 known ✓ Q92731 1/20 0.42
HDAC8 known ✓ Q9BY41 1/20 0.42
ALOX5 known ✓ P09917 1/20 0.40
PTGS2 known ✓ P35354 1/20 0.40
CYP1A2 P05177 1/20 0.93
ALDH1A1 P00352 5/20 0.53
ALOX15 P16050 1/20 0.53
HSD17B10 Q99714 2/20 0.48
SELL P14151 1/20 0.48
SELP P16109 1/20 0.48
TSHR P16473 3/20 0.46
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA7 P43166 3/20 0.46
CA9 Q16790 3/20 0.46
CA14 Q9ULX7 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
CASP1 P29466 1/20 0.44
KDM4E B2RXH2 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL7231103 1.00 CYP1A2 (0.93) CYP1A2ALDH1A1ALOX15HSD17B10SELL
SCHEMBL22122 0.97 CYP1A2 (1.00) CYP1A2ALDH1A1ALOX15HSD17B10SELL
SCHEMBL29417502 0.97 CYP1A2 (1.00) CYP1A2ALDH1A1ALOX15HSD17B10SELL
SCHEMBL31441233 0.93 CYP1A2 (0.93) CYP1A2ALDH1A1ALOX15HSD17B10SELL
Lithium SCHEMBL30762268 0.93 CYP1A2 (0.93) CYP1A2ALDH1A1ALOX15HSD17B10SELL
SCHEMBL7737377 0.93 CYP1A2 (0.93) CYP1A2ALDH1A1ALOX15HSD17B10SELL
SCHEMBL268488 0.93 CYP1A2 (0.93) CYP1A2ALDH1A1ALOX15HSD17B10SELL
Hydrochloric Acid SCHEMBL9860390 0.93 CYP1A2 (0.93) CYP1A2ALDH1A1ALOX15HSD17B10SELL
Lithium SCHEMBL30762269 0.93 CYP1A2 (0.93) CYP1A2ALDH1A1ALOX15HSD17B10SELL
Hydrochloric Acid SCHEMBL338127 0.93 CYP1A2 (0.93) CYP1A2ALDH1A1ALOX15HSD17B10SELL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057262-A REACTING A BIOMASS FEEDSTOCK WITH A PROCESSING AGENT IN THE PRESENCE OF AN ACTIVATION AGENT, HEATING THE BIOMASS MIXTURE, LEACHING AND DRYING UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2000-05-02 US claimed
US-5683793-A Ink jet transparencies XEROX CORPORATION (US) 1997-11-04 US claimed
US-5589277-A INK JET PRINTING, AQUEOUS INKS, FAST DRYING XEROX CORPORATION (US) 1996-12-31 US claimed
EP-0667246-A1 Recording sheets containing amino acids, hydroxy acids, and polycarboxyl compounds XEROX CORPORATION (US) 1995-08-16 EP claimed
CN-107043391-B Organic electroluminescent material containing alkaline earth metal-organic framework and device 中央研究院 2019-08-06 CN disclosed
US-9278909-B2 Amide-extended crosslinking compounds and methods for use thereof DESIGNER MOLECULES, INC. (US) 2016-03-08 US disclosed
US-8637611-B2 Amide-extended crosslinking compounds and methods for use thereof DESIGNER MOLECULES, INC. (US) 2014-01-28 US disclosed
US-20130338313-A1 AMIDE-EXTENDED CROSSLINKING COMPOUNDS AND METHODS FOR USE THEREOF DESIGNER MOLECULES, INC. (US) 2013-12-19 US disclosed
US-20130203895-A1 CURING AGENTS FOR EPOXY RESINS DESIGNER MOLECULES, INC. (US) 2013-08-08 US disclosed
US-20130199724-A1 CURATIVES FOR EPOXY COMPOSITIONS DESIGNER MOLECULES, INC. (US) 2013-08-08 US disclosed
US-20130012620-A1 CURING AGENTS FOR EPOXY RESINS DESIGNER MOLECULES, INC. (US) 2013-01-10 US disclosed
US-8288591-B2 Curing agents for epoxy resins DESIGNER MOLECULES, INC. (US) 2012-10-16 US disclosed
US-20040176537-A1 Inherently electrostatic dissipating block copolymer compositions EASTMAN CHEMICAL COMPANY 2004-09-09 US disclosed
US-6667194-B1 Method of bonding die chip with underfill fluxing composition HENKEL LOCTITE CORPORATION 2003-12-23 US disclosed
WO-2003104245-A1 MULTIMER FORMS OF MONO- AND BIS-ACYLPHOSPHINE OXIDES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2003-12-18 WO disclosed
US-20030130419-A1 Inherently electrostatic dissipating block copolymer compositions EASTMAN CHEMICAL COMPANY 2003-07-10 US disclosed
EP-1304355-A2 Inherently electrostatic dissipating block copolymer compositions EASTMAN CHEMICAL COMPANY (US) 2003-04-23 EP disclosed
US-20030035917-A1 Image making medium HYMAN SYDNEY (US) 2003-02-20 US disclosed
US-6110264-A Phase change inks and methods of forming phase change inks XEROX CORPORATION (US) 2000-08-29 US disclosed
US-6057262-A REACTING A BIOMASS FEEDSTOCK WITH A PROCESSING AGENT IN THE PRESENCE OF AN ACTIVATION AGENT, HEATING THE BIOMASS MIXTURE, LEACHING AND DRYING UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2000-05-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130012620-A1 CURING AGENTS FOR EPOXY RESINS DOT1L, EHMT1, ASH1L ESR2 802/4885HDAC8 237/4885ALOX5 59/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.