SCHEMBL7150372

SCHEMBL7150372

Cc1nn2c(=O)c(CCN3CCC(n4ccc5cc(F)ccc54)CC3)c(C)nc2s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 11/20 0.47
HTR7 P34969 5/20 0.47
KCNH2 Q12809 4/20 0.47
CYP2D6 P10635 4/20 0.41
TSHR P16473 4/20 0.41
HTR2C P28335 4/20 0.41
MAPT P10636 3/20 0.41
HTR1A P08908 3/20 0.41
PMP22 Q01453 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
MEN1 O00255 2/20 0.41
CYP3A4 P08684 2/20 0.41
PKM P14618 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 1/20 0.41
THPO P40225 1/20 0.41
DRD2 P14416 10/20 0.40
ADRA2A P08913 3/20 0.40
ADRA2B P18089 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7150378 0.88 HTR2A (0.47) HTR2AHTR7KCNH2CYP2D6TSHR
SCHEMBL7142123 0.84 HTR2A (0.59) HTR2AHTR7KCNH2CYP2D6TSHR
SCHEMBL7145886 0.80 HTR2A (0.47) HTR2AHTR7KCNH2CYP2D6TSHR
SCHEMBL7140214 0.79 HTR2A (0.61) HTR2AHTR7KCNH2CYP2D6TSHR
SCHEMBL10920489 0.78 HTR2C (0.64) HTR2AHTR7CYP2D6TSHRHTR2C
SCHEMBL7147314 0.71 CYP2D6 (0.54) HTR2AHTR7CYP2D6TSHRHTR2C
SCHEMBL7150338 0.70 DRD2 (0.51) HTR2AHTR7CYP2D6TSHRHTR2C
SCHEMBL8473649 0.70 HTR2A (0.42) HTR2AHTR7KCNH2MAPTHTR1A
SCHEMBL7145335 0.69 DRD2 (0.52) HTR2AHTR7CYP2D6TSHRHTR2C
SCHEMBL10948649 0.68 ADRA1D (0.48) HTR2AHTR7KCNH2DRD2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808313-B1 ANTIPSYCHOTIC 4-(1H-INDOLYL-1-YL)-1-SUBSTITUTED PIPERIDINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2003-08-13 EP disclosed
US-5919788-A PSYCHOLOGICAL DISORDERS JANSSEN PHARMACEUTICA, N.V. (BE) 1999-07-06 US disclosed