SCHEMBL7154140

SCHEMBL7154140

CCc1n[c]cn1-c1cccc(OC(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.47
RXRA P19793 10/20 0.43
GRIN1 Q05586 10/20 0.43
GRIN2B Q13224 10/20 0.43
PIM1 P11309 1/20 0.39
PDE10A Q9Y233 1/20 0.37
DHFR P00374 1/20 0.36
PPARG P37231 1/20 0.36
NOTUM Q6P988 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
CCKAR P32238 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7155477 0.83 KCNH2 (0.42) KCNH2RXRAGRIN1GRIN2BPIM1
SCHEMBL7249466 0.83 ALDH1A1 (0.46) KCNH2DHFRNOTUM
SCHEMBL28266413 0.69 PIM1 (0.46) KCNH2RXRAGRIN1GRIN2BPIM1
SCHEMBL178310 0.69 CHRM2 (0.55) GRIN2B
SCHEMBL28266377 0.69 RXRA (0.47) KCNH2RXRAGRIN1GRIN2BPIM1
SCHEMBL7163341 0.69 MAPT (0.37) KCNH2
SCHEMBL8829657 0.68 RXRA (0.42) KCNH2RXRAGRIN1GRIN2BPIM1
SCHEMBL8139457 0.68 KCNH2 (0.43) KCNH2RXRAGRIN1GRIN2BPDE10A
SCHEMBL21863291 0.68 RXRA (0.73) KCNH2RXRAGRIN1GRIN2BNOTUM
Hydrochloric Acid SCHEMBL21272596 0.66 CHRM2 (0.52) GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358165-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-05 EP disclosed
WO-2002060877-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-08 WO disclosed