SCHEMBL7159796

SCHEMBL7159796

COc1cccc(CCC(N)[C@@H](O)[C@@H](N)Cc2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.52
AOC3 Q16853 1/20 0.49
ABCB1 P08183 3/20 0.46
HTR1A P08908 2/20 0.46
DRD2 P14416 2/20 0.46
SLC2A1 P11166 1/20 0.45
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
METAP2 P50579 1/20 0.44
METAP1 P53582 1/20 0.44
CYP2D6 P10635 2/20 0.44
HTR2A P28223 2/20 0.44
IDO1 P14902 1/20 0.43
AGXT P21549 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7048503 0.83 CAPN1 (0.51) TAAR1AOC3HTR2A
SCHEMBL7051572 0.80 TAAR1 (0.46) TAAR1METAP2METAP1IDO1AGXT
SCHEMBL7050872 0.80 IDO1 (0.50) TAAR1AOC3METAP2IDO1
SCHEMBL3353932 0.78 BCHE (0.52) TAAR1SLC2A1CHRM2CHRM1CHRM3
Hydrochloric Acid SCHEMBL5225498 0.77 BCHE (0.51) TAAR1SLC2A1CHRM2CHRM1CHRM3
SCHEMBL5246588 0.76 TAAR1 (0.69) TAAR1SLC2A1CYP2D6IDO1AGXT
SCHEMBL7047857 0.76 METAP2 (0.52) TAAR1METAP2METAP1
SCHEMBL7713131 0.76 TAAR1 (0.57) TAAR1AOC3ABCB1HTR1ADRD2
SCHEMBL30849685 0.76 TAAR1 (0.53) TAAR1AOC3ABCB1HTR1ADRD2
SCHEMBL7710830 0.76 TAAR1 (0.53) TAAR1AOC3ABCB1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004502669-A 2004-01-29 JP claimed
EP-1353898-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2003-10-22 EP claimed
WO-2002002512-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2002-01-10 WO claimed