SCHEMBL7161306

SCHEMBL7161306

COc1cc(C(O)c2c[nH]cn2)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.38
DYRK1A Q13627 1/20 0.36
MAPK1 P28482 2/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 2/20 0.36
NFKB1 P19838 1/20 0.35
CNR2 P34972 1/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
KMO O15229 1/20 0.34
GRM4 Q14833 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
BLM P54132 1/20 0.34
PMP22 Q01453 1/20 0.34
MEN1 O00255 1/20 0.34
PKM P14618 1/20 0.34
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7159601 0.89 ACHE (0.38) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL7228596 0.84 ACHE (0.38) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL7159560 0.81 ROCK2 (0.38) ACHEMAPK1LMNAGAAHTT
SCHEMBL7098179 0.81 ALDH1A1 (0.38) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL6784764 0.79 S1PR1 (0.36) GAAHTTSMN1; SMN2KMT2AKMO
SCHEMBL6929116 0.77 CASR (0.39) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL7104909 0.76 GRM8 (0.43) HTTSMN1; SMN2KMT2AGRM4PKM
SCHEMBL7247069 0.74 ADRB3 (0.43) MAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL21624997 0.74 CHEK2 (0.35)
SCHEMBL632963 0.73 DYRK1A (0.36) DYRK1AMAPK1KMT2ANFKB1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358165-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-05 EP disclosed
WO-2002060877-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-08 WO disclosed