SCHEMBL7228596

SCHEMBL7228596

COc1cc(C(O)c2c[nH]cn2)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.38
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NFKB1 P19838 1/20 0.35
BLM P54132 2/20 0.34
PMP22 Q01453 1/20 0.34
GRM4 Q14833 1/20 0.34
KMT2A Q03164 1/20 0.33
TSHR P16473 2/20 0.33
CYP3A4 P08684 1/20 0.33
PPARG P37231 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33
IDH1 O75874 1/20 0.32
CNR2 P34972 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GRM2 Q14416 1/20 0.32
GRM3 Q14832 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7159560 0.89 ROCK2 (0.38) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL7161306 0.84 ACHE (0.38) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL7159601 0.81 ACHE (0.38) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL7098179 0.81 ALDH1A1 (0.38) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL7162387 0.79 RXRA (0.30)
SCHEMBL6929116 0.77 CASR (0.39) ACHELMNAGAAHTTSMN1; SMN2
SCHEMBL7104909 0.76 GRM8 (0.43) HTTSMN1; SMN2GRM4KMT2ATSHR
SCHEMBL7247069 0.74 ADRB3 (0.43) SMN1; SMN2KMT2A
SCHEMBL7158323 0.74 PDE2A (0.38)
SCHEMBL21624997 0.74 CHEK2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667335-B2 NMDA (N-methyl-D-aspartate)-receptor subtype selective blockers HOFFMANN-LA ROCHE INC. 2003-12-23 US disclosed