SCHEMBL716840

SCHEMBL716840

CS(=O)(=O)CNc1cc(C(=O)O)cc(C(=O)N2CCCC2c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
RIPK1 Q13546 1/20 0.45
SCD O00767 3/20 0.44
SCD5 Q86SK9 5/20 0.43
KCNK3 O14649 1/20 0.43
ROCK2 O75116 3/20 0.42
EPHX2 P34913 2/20 0.41
PARP14 Q460N5 1/20 0.41
PARP10 Q53GL7 1/20 0.41
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
PPID Q08752 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL717696 0.91 RIPK1 (0.45) HSP90AA1HSP90AB1RIPK1SCDSCD5
SCHEMBL715644 0.85 POLB (0.50)
SCHEMBL175220 0.82 HSP90AA1 (0.46) HSP90AA1HSP90AB1RIPK1SCDSCD5
SCHEMBL715025 0.80 NAA50 (0.38)
SCHEMBL166963 0.80 RIPK1 (0.54) HSP90AA1HSP90AB1RIPK1SCDSCD5
SCHEMBL167323 0.79 HSP90AA1 (0.47) HSP90AA1HSP90AB1RIPK1SCDSCD5
SCHEMBL716612 0.76 NPC1 (0.46)
SCHEMBL164387 0.76 PARP14 (0.60) HSP90AA1HSP90AB1RIPK1SCDSCD5
SCHEMBL256556 0.72 RIPK1 (0.53) HSP90AA1HSP90AB1RIPK1SCDSCD5
SCHEMBL256561 0.72 HSP90AA1 (0.46) HSP90AA1HSP90AB1RIPK1SCDSCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120053200-A1 BACE 2 INHIBITORS HOFFMANN-LA ROCHE INC. 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053200-A1 BACE 2 INHIBITORS BACE2, BACE1, PSEN2 HSP90AA1 3048/4885HSP90AB1 1398/4885RIPK1 3784/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.