SCHEMBL7170644

SCHEMBL7170644

COC(=O)N1C[C@@H]2CCC(CNC(C)(C#N)c3cccc4ccccc34)CC2CC1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.31
PREP P48147 3/20 0.31
ACKR3 P25106 1/20 0.30
FAP Q12884 1/20 0.30
LTC4S Q16873 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7162414 0.80 DPP4 (0.41) DPP4
SCHEMBL7170649 0.75 LTC4S (0.37) DPP4PREPFAPLTC4S
SCHEMBL7171997 0.74 CXCR4 (0.40) DPP4
SCHEMBL7165958 0.73 AGTR2 (0.41) DPP4
SCHEMBL7170826 0.71 CXCR4 (0.40)
SCHEMBL7168153 0.70 GRIN2B (0.46)
SCHEMBL7163823 0.70 PGR (0.40) DPP4FAP
SCHEMBL7166169 0.70 CXCR4 (0.43)
SCHEMBL7161639 0.70 PGR (0.35)
SCHEMBL7168130 0.69 KMT2A (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003082856-A1 ISOQUINOLINE-3-CARBOXYLIC ACID DERIVATIVES AS EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2003-10-09 WO disclosed