SCHEMBL7170649

SCHEMBL7170649

COC(=O)N1C[C@@H]2CCC(CN(CC#N)Cc3cccc4ccccc34)CC2CC1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LTC4S Q16873 4/20 0.37
DPP4 P27487 1/20 0.35
HTT P42858 1/20 0.33
PREP P48147 4/20 0.32
ACE P12821 1/20 0.31
FAP Q12884 1/20 0.31
GRIK1 P39086 1/20 0.31
P2RX7 Q99572 1/20 0.31
GRM2 Q14416 1/20 0.31
GRM3 Q14832 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7169997 0.89 SMN1; SMN2 (0.37)
SCHEMBL7161639 0.88 PGR (0.35) ACE
SCHEMBL7163823 0.87 PGR (0.40) DPP4FAP
SCHEMBL7141654 0.83 LTC4S (0.37) LTC4S
SCHEMBL7166478 0.83 AGTR2 (0.37) ACE
SCHEMBL7170300 0.83 TAS2R14 (0.35) LTC4S
SCHEMBL7162414 0.81 DPP4 (0.41) DPP4HTTP2RX7GRM2GRM3
SCHEMBL7170644 0.75 DPP4 (0.31) LTC4SDPP4PREPFAP
SCHEMBL7170826 0.71 CXCR4 (0.40) ACEP2RX7
SCHEMBL7168153 0.70 GRIN2B (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003082856-A1 ISOQUINOLINE-3-CARBOXYLIC ACID DERIVATIVES AS EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2003-10-09 WO disclosed