SCHEMBL7192028

SCHEMBL7192028

N=[N+]=C(C(=O)C[C@@H]1CN(C(=O)[O-])[C@@H]2C(=O)N[C@H]12)C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 2/20 0.36
ATM Q13315 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9705614 0.84 TDP1 (0.39) TDP1ALDH1A1ATMMAPTHPGD
SCHEMBL7186704 0.84 TDP1 (0.39) TDP1ALDH1A1ATMMAPTHPGD
SCHEMBL9032259 0.80 TDP1 (0.38) TDP1ALDH1A1ATMMAPTHPGD
SCHEMBL9871979 0.69 TDP1 (0.41) TDP1ALDH1A1ATMMAPTHPGD
SCHEMBL22581180 0.64 HTR2A (0.40) TDP1ALDH1A1MAPTHPGDRAB9A
SCHEMBL9168542 0.64 RAB9A (0.35) TDP1ATMRAB9APOLBSMN1; SMN2
SCHEMBL10493918 0.64 ALDH1A1 (0.37) ALDH1A1MAPTHPGDRAB9APOLB
SCHEMBL9670137 0.64 ALDH1A1 (0.39) TDP1ALDH1A1MAPTHPGDRAB9A
SCHEMBL2944429 0.64 RAB9A (0.35) TDP1ATMRAB9APOLBSMN1; SMN2
SCHEMBL10790770 0.64 RAB9A (0.35) TDP1ATMRAB9APOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6566355-B1 Useful in combination with beta -lactam antibiotics in the control of beta -lactamase forming pathogens HOFFMANN-LA ROCHE INC. 2003-05-20 US disclosed