SCHEMBL7196147

SCHEMBL7196147

CN1C(=O)C(NC(=O)OCc2ccccc2)NC(=O)C2=C1CCC=C2

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
NAAA Q02083 1/20 0.39
TSHR P16473 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CTSB P07858 3/20 0.37
CTSK P43235 3/20 0.37
CTSL P07711 2/20 0.37
CPB1 P15086 1/20 0.37
TLR4 O00206 1/20 0.37
PREP P48147 2/20 0.37
CTSS P25774 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12879744 0.80 MEN1 (0.48) ALDH1A1GAANAAATSHRMEN1
SCHEMBL7196152 0.78 ALDH1A1 (0.41) ALDH1A1GAANAAATSHRMEN1
SCHEMBL4697243 0.77 SCN9A (0.50) ALDH1A1GAA
SCHEMBL7807139 0.68 GAA (0.44) ALDH1A1GAANAAATSHRCTSB
SCHEMBL7807134 0.68 GAA (0.44) ALDH1A1GAANAAATSHRCTSB
SCHEMBL12345121 0.67 NAAA (0.50) ALDH1A1GAANAAATSHRCTSB
SCHEMBL13017770 0.67 NAAA (0.50) ALDH1A1GAANAAATSHRCTSB
SCHEMBL2010782 0.66 NAAA (0.55) ALDH1A1GAANAAATSHRCTSB
SCHEMBL19576597 0.66 ALDH1A1 (0.53) ALDH1A1GAANAAATSHRCTSB
SCHEMBL33525492 0.66 ALDH1A1 (0.50) ALDH1A1GAANAAATSHRCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294702-A1 BENZODIAZEPINE DERIVATIVES AS APP MODULATORS MERCK SHARP & DOHME LTD. (GB) 2003-03-26 EP disclosed
WO-2001090084-A1 BENZODIAZEPINE DERIVATIVES AS APP MODULATORS MERCK SHARP & DOHME LIMITED (GB) 2001-11-29 WO disclosed