SCHEMBL7807134

SCHEMBL7807134

CN1CCCN[C@@H](NC(=O)OCc2ccccc2)C1=O

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CTSL P07711 1/20 0.44
CTSB P07858 1/20 0.44
CTSK P43235 1/20 0.44
PREP P48147 4/20 0.43
NAAA Q02083 1/20 0.43
TSHR P16473 1/20 0.43
DPP4 P27487 1/20 0.43
KCNH2 Q12809 1/20 0.43
DPP7 Q9UHL4 1/20 0.43
EPHX1 P07099 1/20 0.43
CPB1 P15086 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7807139 1.00 GAA (0.44) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL13043811 0.80 CASP3 (0.53) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL14337553 0.80 CASP3 (0.53) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL7811138 0.79 ALDH1A1 (0.45) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL7811136 0.79 ALDH1A1 (0.45) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL6199396 0.77 NAAA (0.51) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL21111192 0.77 CPB1 (0.49) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL13043801 0.77 CTSK (0.54) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL14601914 0.77 CTSK (0.54) GAAALDH1A1CTSLCTSBCTSK
SCHEMBL12879744 0.76 MEN1 (0.48) GAAALDH1A1PREPNAAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855397-B1 (R)-5-BROMO-N-(1-ETHYL-4-METHYLHEXAHYDRO-1H-1,4-DIAZEPIN-6-YL)-2-METHOXY-6-METHYLAMINO-3-PYRIDINE-CARBOXAMIDE, PROCESS FOR PRODUCING THE SAME AND MEDICINAL COMPOSITION CONTAINING THE SAME DAINIPPON PHARMACEUTICAL CO (JP) 2001-05-09 EP disclosed
US-5945415-A GASTROINTESTINAL DISORDERS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1999-08-31 US disclosed
EP-0855397-A1 (R)-5-BROMO-N-(1-ETHYL-4-METHYLHEXAHYDRO-1H-1,4-DIAZEPIN-6-YL)-2-METHOXY-6-METHYLAMINO-3-PYRIDINE-CARBOXAMIDE, PROCESS FOR PRODUCING THE SAME AND MEDICINAL COMPOSITION CONTAINING THE SAME DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1998-07-29 EP disclosed