SCHEMBL7196152

SCHEMBL7196152

CN1C(=O)C(NC(=O)OCc2ccccc2)NC(=O)C2=CCCC=C21

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
CPB1 P15086 1/20 0.41
CTSB P07858 3/20 0.40
CTSK P43235 3/20 0.40
CTSS P25774 2/20 0.40
CTSL P07711 2/20 0.40
NAAA Q02083 1/20 0.40
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PREP P48147 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ADORA1 P30542 1/20 0.38
ADORA2B P29275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12879744 0.81 MEN1 (0.48) ALDH1A1GAACPB1NAAATSHR
SCHEMBL4697243 0.79 SCN9A (0.50) ALDH1A1GAA
SCHEMBL7196147 0.78 ALDH1A1 (0.39) ALDH1A1GAACPB1CTSBCTSK
SCHEMBL7807134 0.69 GAA (0.44) ALDH1A1GAACPB1CTSBCTSK
SCHEMBL7807139 0.69 GAA (0.44) ALDH1A1GAACPB1CTSBCTSK
SCHEMBL13017770 0.69 NAAA (0.50) ALDH1A1GAACTSBCTSLNAAA
SCHEMBL12345121 0.69 NAAA (0.50) ALDH1A1GAACTSBCTSLNAAA
SCHEMBL7811138 0.67 ALDH1A1 (0.45) ALDH1A1GAACPB1CTSBCTSK
SCHEMBL12527905 0.67 CASP3 (0.49) ALDH1A1GAACTSBCTSKCTSS
SCHEMBL9541279 0.67 ALDH1A1 (0.52) ALDH1A1GAACPB1CTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294702-A1 BENZODIAZEPINE DERIVATIVES AS APP MODULATORS MERCK SHARP & DOHME LTD. (GB) 2003-03-26 EP disclosed
WO-2001090084-A1 BENZODIAZEPINE DERIVATIVES AS APP MODULATORS MERCK SHARP & DOHME LIMITED (GB) 2001-11-29 WO disclosed